| Assay ID | Title | Year | Journal | Article |
|---|
| AID1347154 | Primary screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1508630 | Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident proteome: Secreted ER Calcium Modulated Protein (SERCaMP) assay | 2021 | Cell reports, 04-27, Volume: 35, Issue:4
| A target-agnostic screen identifies approved drugs to stabilize the endoplasmic reticulum-resident proteome. |
| AID1345685 | Human A1 receptor (Adenosine receptors) | 2002 | Journal of medicinal chemistry, Mar-28, Volume: 45, Issue:7
| 1,8-disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists. |
| AID1345690 | Rat A2A receptor (Adenosine receptors) | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID1345721 | Human A2B receptor (Adenosine receptors) | 2002 | Journal of medicinal chemistry, Mar-28, Volume: 45, Issue:7
| 1,8-disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists. |
| AID1345822 | Human A3 receptor (Adenosine receptors) | 2002 | Journal of medicinal chemistry, Mar-28, Volume: 45, Issue:7
| 1,8-disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists. |
| AID1345630 | Rat A1 receptor (Adenosine receptors) | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID1289959 | Displacement of [3H]ZM241385 from human recombinant Adenosine A2B receptor | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes. |
| AID267463 | Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cells | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| AID1549354 | Displacement of [3H]NECA from recombinant mouse A3 adenosine receptor expressed in CHO cell membranes measured after 180 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1851393 | Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane and measured after 0.5 hrs by radioligand displacement assay | 2022 | RSC medicinal chemistry, Jul-20, Volume: 13, Issue:7
| Development of subtype-selective covalent ligands for the adenosine A |
| AID30807 | Binding affinity against Adenosine A2 receptor in rat striatal membranes using [3H]5'-(N-ethylcarboxamido)-adenosine (NECA) as the ligand | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID1549355 | Displacement of [3H]ZM241385 from recombinant human A2B adenosine receptor expressed in CHO cell membranes measured after 30 mins by scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1549357 | Displacement of [3H]CCPA from recombinant human A1 adenosine receptor expressed in CHO cell membranes measured after 20 hrs by microplate filtration based radioligand binding assay | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1744261 | Antagonist activity at human A2B receptor | 2021 | Journal of medicinal chemistry, 01-14, Volume: 64, Issue:1
| 3,4-Dihydropyrimidin-2(1 |
| AID1549319 | Displacement of [3H]DPCPX from recombinant mouse A1 adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1549350 | Binding affinity to rat A3 adenosine receptor | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1549351 | Displacement of [3H]PSB-603 from recombinant mouse A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID32867 | Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranes | 2004 | Journal of medicinal chemistry, Feb-12, Volume: 47, Issue:4
| Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability. |
| AID34727 | Binding affinity for human adenosine A3 receptor using [3H]PBS-11 in CHO cell membranes; ND denotes not determined | 2004 | Journal of medicinal chemistry, Feb-12, Volume: 47, Issue:4
| Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability. |
| AID1851395 | Ratio of Ki for displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane to Ki for displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4hrs | 2022 | RSC medicinal chemistry, Jul-20, Volume: 13, Issue:7
| Development of subtype-selective covalent ligands for the adenosine A |
| AID1851403 | Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane assessed as covalent adduct formation at 10 uM preincubated followed by 4 times washing treatment and then with [3H]PSB-603 exposure by radioligand displacement a | 2022 | RSC medicinal chemistry, Jul-20, Volume: 13, Issue:7
| Development of subtype-selective covalent ligands for the adenosine A |
| AID1549361 | Displacement of [3H]CCPA from A1 adenosine receptor in rat cortex membranes measured after 60 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID267466 | Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in CHO cells | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| AID1549360 | Displacement of [3H]NECA from rat A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID1549358 | Displacement of [3H]PSB-11 from recombinant human A3 adenosine receptor expressed in CHO cell membranes by radioligand binding assay | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID31881 | Binding affinity at Adenosine A1 receptor in rat brain cortical membrane using [3H]N6-R-phenylisopropyladenosine (R-PIA) as radioligand | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID1549352 | Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID267462 | Displacement of [3H]R-PIA from adenosine A2A receptor in rat brain striatal membranes | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| AID1549356 | Displacement of [3H]MSX-2 from recombinant human A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID32045 | Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparations | 2004 | Journal of medicinal chemistry, Feb-12, Volume: 47, Issue:4
| Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability. |
| AID1549359 | Displacement of [3H]PSB-603 from recombinant rat A2B adenosine receptor expressed in CHO cell membranes measured after 75 mins by liquid scintillation counting method | 2019 | Journal of medicinal chemistry, 04-25, Volume: 62, Issue:8
| A |
| AID33286 | Binding affinity for human adenosine A2B receptor using [3H]PSB-298 in CHO cell membranes; ND denotes not determined | 2004 | Journal of medicinal chemistry, Feb-12, Volume: 47, Issue:4
| Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability. |
| AID267460 | Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| AID267467 | Displacement of [3H]PSB11 from human recombinant adenosine A3 receptor expressed in CHO cells | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| AID1482184 | Displacement of [3H]ZM241385 from human recombinant adenosine A2B receptor | 2017 | Journal of medicinal chemistry, 04-27, Volume: 60, Issue:8
| Enantiospecific Recognition at the A |
| AID1851394 | Displacement of [3H]PSB-603 from human adenosine A2B receptor expressed in CHO cell membrane preincubated for 4 hrs followed by [3H]PSB-603 addition and measured after 0.5 hrs by radioligand displacement assay | 2022 | RSC medicinal chemistry, Jul-20, Volume: 13, Issue:7
| Development of subtype-selective covalent ligands for the adenosine A |
| AID267459 | Displacement of [3H]R-PIA from adenosine A1 receptor in rat brain cortical membranes | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |