| Assay ID | Title | Year | Journal | Article |
|---|
| AID32643 | Relative affinities for rat Adenosine A1 and Adenosine A2B receptors | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID32017 | Binding affinity of [3H]R-PIA for rat Adenosine A2B receptor in HEK293 cells | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID33579 | Binding affinity to A2 adenosine receptor from rat striatal membrane in presence of [3H]5'-(N-ethylcarboximido)-adenosine | 1994 | Journal of medicinal chemistry, May-13, Volume: 37, Issue:10
| Synthesis and structure-activity relationships of deazaxanthines: analogs of potent A1- and A2-adenosine receptor antagonists. |
| AID74022 | Relaxant activity on the spontaneous tone of isolated guinea pig tracheal ring chains. | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID33021 | Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatal membranes | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID34705 | Inhibition of [125I]I-AB-MECA binding to human Adenosine A3 receptor | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID30500 | Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPX | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID227877 | Ratio of stimulatory activity in right atrium to relaxant activity in tracheal muscle | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID30807 | Binding affinity against Adenosine A2 receptor in rat striatal membranes using [3H]5'-(N-ethylcarboxamido)-adenosine (NECA) as the ligand | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID33176 | Binding affinity at human Adenosine A2B receptor expressed in HEK293 cells, using [125I]ABOPX as radioligand | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID32642 | Relative affinities for rat Adenosine A1 and Adenosine A2B receptors | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| AID75917 | Positive chronotropic effect on isolated guinea pig right atrium (heart stimulation). | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID32155 | Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]CPX. | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID219846 | Inhibition of c-AMP phosphodiesterase activity in guinea pig tracheal muscle | 1992 | Journal of medicinal chemistry, Oct-30, Volume: 35, Issue:22
| Effects of alkyl substitutions of xanthine skeleton on bronchodilation. |
| AID227036 | A1 selectivity is the ratio between A2 and A1 receptor | 1994 | Journal of medicinal chemistry, May-13, Volume: 37, Issue:10
| Synthesis and structure-activity relationships of deazaxanthines: analogs of potent A1- and A2-adenosine receptor antagonists. |
| AID31881 | Binding affinity at Adenosine A1 receptor in rat brain cortical membrane using [3H]N6-R-phenylisopropyladenosine (R-PIA) as radioligand | 1993 | Journal of medicinal chemistry, Oct-29, Volume: 36, Issue:22
| Synthesis of paraxanthine analogs (1,7-disubstituted xanthines) and other xanthines unsubstituted at the 3-position: structure-activity relationships at adenosine receptors. |
| AID32039 | Binding affinity to A1 adenosine receptor from rat cortical membrane in presence of [3H]R-(phenylisopropyl)-adenosine | 1994 | Journal of medicinal chemistry, May-13, Volume: 37, Issue:10
| Synthesis and structure-activity relationships of deazaxanthines: analogs of potent A1- and A2-adenosine receptor antagonists. |
| AID33610 | Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cells | 2002 | Journal of medicinal chemistry, May-23, Volume: 45, Issue:11
| Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |