Page last updated: 2024-08-07 18:44:20
Adenosine receptor A2a
An adenosine receptor A2a that is encoded in the genome of mouse. [OMA:Q60613, PRO:DNx]
Synonyms
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 2 (66.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosine | Mus musculus (house mouse) | Ki | 1.0000 | 1 | 1 |
2-chloro-n(6)cyclopentyladenosine | Mus musculus (house mouse) | Ki | 0.9880 | 1 | 1 |
n(6)-cyclopentyladenosine | Mus musculus (house mouse) | Ki | 0.8080 | 1 | 1 |
2-chloro-n(6)-(3-iodobenzyl)adenosine-5'-n-methyluronamide | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
psb 1115 | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
mrs 1754 | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
mrs 3558 | Mus musculus (house mouse) | Ki | 10.4000 | 1 | 1 |