Page last updated: 2024-08-07 23:57:06
Adenosine receptor A3
An adenosine receptor A3 that is encoded in the genome of mouse. [OMA:Q61618, PRO:WCB]
Synonyms
A3AR
Research
Bioassay Publications (7)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (14.29) | 29.6817 |
| 2010's | 4 (57.14) | 24.3611 |
| 2020's | 2 (28.57) | 2.80 |
Compounds (11)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosine | Mus musculus (house mouse) | Ki | 0.0001 | 1 | 1 |
| 2-chloro-n(6)cyclopentyladenosine | Mus musculus (house mouse) | Ki | 0.0170 | 1 | 1 |
| adenosine-5'-(n-ethylcarboxamide) | Mus musculus (house mouse) | Ki | 0.0141 | 1 | 1 |
| n(6)-cyclopentyladenosine | Mus musculus (house mouse) | Ki | 0.5340 | 1 | 1 |
| 2-chloro-n(6)-(3-iodobenzyl)adenosine-5'-n-methyluronamide | Mus musculus (house mouse) | Ki | 0.0002 | 1 | 1 |
| mrs 1523 | Mus musculus (house mouse) | Ki | 0.3490 | 1 | 1 |
| mre 3008-f20 | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| psb 1115 | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| mrs 1754 | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| mrs 3558 | Mus musculus (house mouse) | Ki | 0.0015 | 1 | 1 |
| psb 11 | Mus musculus (house mouse) | Ki | 6.3600 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| adenosine-5'-(n-ethylcarboxamide) | Mus musculus (house mouse) | EC50 | 0.1880 | 1 | 1 |
| 2-chloro-n(6)-(3-iodobenzyl)adenosine-5'-n-methyluronamide | Mus musculus (house mouse) | EC50 | 0.0003 | 2 | 2 |