| Assay ID | Title | Year | Journal | Article |
|---|
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1180477 | Inhibition of rat MAO-A in rat-liver mitochondrial-fraction using [14C]-5-HT substrate | 2014 | Journal of medicinal chemistry, Aug-14, Volume: 57, Issue:15
| Indazole- and indole-5-carboxamides: selective and reversible monoamine oxidase B inhibitors with subnanomolar potency. |
| AID1657005 | Inhibition of acetylcholinesterase (unknown origin) | 2020 | Journal of medicinal chemistry, 06-11, Volume: 63, Issue:11
| Acetylene Group, Friend or Foe in Medicinal Chemistry. |
| AID1657006 | Inhibition of butyrylcholinesterase (unknown origin) | 2020 | Journal of medicinal chemistry, 06-11, Volume: 63, Issue:11
| Acetylene Group, Friend or Foe in Medicinal Chemistry. |
| AID126214 | Inhibitory activity against Monoamine oxidase A | 2000 | Journal of medicinal chemistry, May-04, Volume: 43, Issue:9
| Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition. |
| AID1195745 | Selectivity ratio of IC50 for human MAO-A expressed in baculovirus infected BTI insect cells to IC50 for human MAO-B expressed in baculovirus infected BTI insect cells | 2014 | Journal of medicinal chemistry, Dec-26, Volume: 57, Issue:24
| N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor. |
| AID1657003 | Inhibition of Sprague-Dawley rat liver mitochondrial MAO-A using [14C]-5-HT as substrate after 30 mins by liquid scintillation counting | 2020 | Journal of medicinal chemistry, 06-11, Volume: 63, Issue:11
| Acetylene Group, Friend or Foe in Medicinal Chemistry. |
| AID127191 | Inhibitory activity against Monoamine oxidase B | 2000 | Journal of medicinal chemistry, May-04, Volume: 43, Issue:9
| Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition. |
| AID1180478 | Inhibition of rat MAO-B in rat-liver mitochondrial-fraction using [14C]-PEA substrate | 2014 | Journal of medicinal chemistry, Aug-14, Volume: 57, Issue:15
| Indazole- and indole-5-carboxamides: selective and reversible monoamine oxidase B inhibitors with subnanomolar potency. |
| AID127172 | Inhibitory activity against Monoamine oxidase B | 2000 | Journal of medicinal chemistry, May-04, Volume: 43, Issue:9
| Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition. |
| AID1195741 | Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells preincubated for 15 mins | 2014 | Journal of medicinal chemistry, Dec-26, Volume: 57, Issue:24
| N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor. |
| AID1195740 | Inhibition of human MAO-A expressed in baculovirus infected BTI insect cells preincubated for 15 mins | 2014 | Journal of medicinal chemistry, Dec-26, Volume: 57, Issue:24
| N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor. |
| AID1657004 | Inhibition of Sprague-Dawley rat liver mitochondrial MAO-B using [14C]-PEA as substrate after 30 mins by liquid scintillation counting | 2020 | Journal of medicinal chemistry, 06-11, Volume: 63, Issue:11
| Acetylene Group, Friend or Foe in Medicinal Chemistry. |
| AID126350 | Inhibitory activity against Monoamine oxidase A | 2000 | Journal of medicinal chemistry, May-04, Volume: 43, Issue:9
| Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |