| Assay ID | Title | Year | Journal | Article |
|---|
| AID30445 | Binding affinity against human adenosine A1 receptor expressed in CHO cells using [3H]DPCPX | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID1874237 | Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance assay | 2022 | ACS medicinal chemistry letters, Jul-14, Volume: 13, Issue:7
| Surface Plasmon Resonance Screening to Identify Active and Selective Adenosine Receptor Binding Fragments. |
| AID1857146 | Displacement of [3H]-DPCPX from human adenosine A1R expressed in CHO cells membrane assessed as dissociation constant (koff) preincubated for 1 hr followed by compound addition and measured after 1 hr | | | |
| AID33951 | Stimulation of human adenosine A2B receptor in production of cAMP in CHO cells | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID34271 | Inhibition of human adenosine A3 receptor in production of cAMP in CHO cells | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID1874235 | Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as affinity on-rate by surface plasmon resonance assay | 2022 | ACS medicinal chemistry letters, Jul-14, Volume: 13, Issue:7
| Surface Plasmon Resonance Screening to Identify Active and Selective Adenosine Receptor Binding Fragments. |
| AID30298 | Inhibition of human adenosine A1 receptor in production of cAMP in CHO cells | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID33617 | Stimulation of human adenosine A2A receptor in production of cAMP in CHO cells | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID1874238 | Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance assay | 2022 | ACS medicinal chemistry letters, Jul-14, Volume: 13, Issue:7
| Surface Plasmon Resonance Screening to Identify Active and Selective Adenosine Receptor Binding Fragments. |
| AID1874236 | Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as affinity off-rate by surface plasmon resonance assay | 2022 | ACS medicinal chemistry letters, Jul-14, Volume: 13, Issue:7
| Surface Plasmon Resonance Screening to Identify Active and Selective Adenosine Receptor Binding Fragments. |
| AID1857145 | Displacement of [3H]-DPCPX from human adenosine A1R expressed in CHO cells membrane assessed as association constant (kon) incubated for 45 mins | | | |
| AID34579 | Binding affinity against human adenosine A3 receptor expressed on HEK293 cells using [125I]I-AB-MECA | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID33950 | Agonistic activity against human adenosine A2B receptor expressed in CHO cells | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| AID1857147 | Displacement of [3H]-DPCPX from human adenosine A1R expressed in CHO cells membrane incubated for 1 hr | | | |
| AID1857148 | Displacement of [3H]-DPCPX from human adenosine A1R expressed in CHO cells membrane assessed as residence time | | | |
| AID33621 | Binding affinity against human adenosine A2A receptor expressed in HEK293 cells using [3H]ZM-241385 | 2004 | Journal of medicinal chemistry, Jul-15, Volume: 47, Issue:15
| New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |