luf-5834 has been researched along with regadenoson* in 1 studies
1 other study(ies) available for luf-5834 and regadenoson
Article | Year |
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A
In drug design, G protein-coupled receptor (GPCR) partial agonists enable one to fine-tune receptor output between basal and maximal signaling levels. Here, we add to the structural basis for rationalizing and monitoring partial agonism. NMR spectroscopy of partial agonist complexes of the A Topics: Adenosine A2 Receptor Agonists; Aminopyridines; Binding Sites; Cell Line; Drug Partial Agonism; Humans; Imidazoles; Molecular Dynamics Simulation; Protein Binding; Purines; Pyrazoles; Receptor, Adenosine A2A | 2021 |