| Assay ID | Title | Year | Journal | Article |
|---|
| AID734064 | Inhibition of human recombinant MMP1 catalytic domain using Dnp-Pro-beta-cyclohexyl-Ala-Gly-Cys(Me)-His-Lys-(Nma)-NH2 as substrate preincubated with enzyme for 30 mins prior to substrate addition measured after 20 mins by fluorometric assay | 2013 | European journal of medicinal chemistry, Apr, Volume: 62 | Synthesis of derivatives of methyl rosmarinate and their inhibitory activities against matrix metalloproteinase-1 (MMP-1). |
| AID307317 | Inhibition of Jurkat cell activation assessed as blocking of T-cell antigen receptor-induced IL-2 expression at 30 uM by luciferase assay | 2007 | Bioorganic & medicinal chemistry, Jun-01, Volume: 15, Issue:11
| The structure-activity relationship of the series of non-peptide small antagonists for p56lck SH2 domain. |
| AID471352 | Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 mins | 2009 | Journal of natural products, Aug, Volume: 72, Issue:8
| Matrix metalloproteinase-2 inhibitors from Clinopodium chinense var. parviflorum. |
| AID670313 | Inhibition of human recombinant MMP9 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID670318 | Inhibition of human recombinant MMP3 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID598345 | Inhibition of TNF-alpha-induced COX2 mRNA expression in human HepG2 cells expressing NF-kappaB preincubated 1 hr before TNFalpha challenge measured after 6 hrs by RT-PCR analysis | 2011 | Bioorganic & medicinal chemistry letters, Jun-01, Volume: 21, Issue:11
| Anti-inflammatory activity of constituents from Glechoma hederacea var. longituba. |
| AID1617647 | Antiinflammatory activity against LPS-stimulated mouse RAW264.7 cells assessed as decrease in PGE2 production preincubated for 1 hr followed by LPS stimulation and measured after 24 hrs by ELISA | | | |
| AID670314 | Inhibition of human recombinant MMP12 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID598309 | Inhibition of TNF-alpha-induced NF-kappaB transactivation expressed in human HepG2 cells at 20 uM preincubated 1 hr before TNFalpha challenge measured after 1 hr by luciferase reporter gene assay | 2011 | Bioorganic & medicinal chemistry letters, Jun-01, Volume: 21, Issue:11
| Anti-inflammatory activity of constituents from Glechoma hederacea var. longituba. |
| AID670317 | Inhibition of human recombinant MMP2 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID670316 | Inhibition of human recombinant MMP1 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID1423273 | Antiproliferative activity against human MV4-11 cells by Cell-Titer Glo assay | 2018 | Journal of natural products, 11-26, Volume: 81, Issue:11
| Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis. |
| AID598311 | Inhibition of TNF-alpha-induced iNOS mRNA expression in human HepG2 cells expressing NF-kappaB preincubated 1 hr before TNFalpha challenge measured after 6 hrs by RT-PCR analysis | 2011 | Bioorganic & medicinal chemistry letters, Jun-01, Volume: 21, Issue:11
| Anti-inflammatory activity of constituents from Glechoma hederacea var. longituba. |
| AID670315 | Inhibition of human recombinant MMP13 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID670320 | Inhibition of human recombinant MMP12 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID1423272 | Antiproliferative activity against human MOLM14 cells by Cell-Titer Glo assay | 2018 | Journal of natural products, 11-26, Volume: 81, Issue:11
| Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis. |
| AID307316 | Inhibition of Jurkat cell activation assessed as blocking of T-cell antigen receptor-induced IL-2 expression at 10 uM by luciferase assay | 2007 | Bioorganic & medicinal chemistry, Jun-01, Volume: 15, Issue:11
| The structure-activity relationship of the series of non-peptide small antagonists for p56lck SH2 domain. |
| AID670319 | Inhibition of human recombinant MMP9 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID670311 | Inhibition of human recombinant MMP2 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID1423271 | Antiproliferative activity against human MOLM13 cells by Cell-Titer Glo assay | 2018 | Journal of natural products, 11-26, Volume: 81, Issue:11
| Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis. |
| AID730190 | Antiviral activity against Respiratory syncytial virus assessed as reduction of virus-induced cytopathic effect at maximal non-toxic concentration | 2013 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 23, Issue:5
| Five new phenolic glycosides from Hedyotis scandens. |
| AID670312 | Inhibition of human recombinant MMP3 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID307315 | Inhibition of p56lck SH2 domain by ELISA | 2007 | Bioorganic & medicinal chemistry, Jun-01, Volume: 15, Issue:11
| The structure-activity relationship of the series of non-peptide small antagonists for p56lck SH2 domain. |
| AID307319 | Partition coefficient, log P of the compound | 2007 | Bioorganic & medicinal chemistry, Jun-01, Volume: 15, Issue:11
| The structure-activity relationship of the series of non-peptide small antagonists for p56lck SH2 domain. |
| AID598307 | Cytotoxicity against human HepG2 cells up to 20 uM after 24 hrs by MTS assay | 2011 | Bioorganic & medicinal chemistry letters, Jun-01, Volume: 21, Issue:11
| Anti-inflammatory activity of constituents from Glechoma hederacea var. longituba. |
| AID734065 | Inhibition of human recombinant MMP1 catalytic domain using Dnp-Pro-beta-cyclohexyl-Ala-Gly-Cys(Me)-His-Lys-(Nma)-NH2 as substrate at 10 uM preincubated with enzyme for 30 mins prior to substrate addition measured after 20 mins by fluorometric assay | 2013 | European journal of medicinal chemistry, Apr, Volume: 62 | Synthesis of derivatives of methyl rosmarinate and their inhibitory activities against matrix metalloproteinase-1 (MMP-1). |
| AID670321 | Inhibition of human recombinant MMP13 catalytic domain at 10 uM incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| AID670310 | Inhibition of human recombinant MMP1 catalytic domain incubated for 20 mins by fluorimetric assay | 2012 | Bioorganic & medicinal chemistry, Jul-01, Volume: 20, Issue:13
| Natural products as a gold mine for selective matrix metalloproteinases inhibitors. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |