| Assay ID | Title | Year | Journal | Article |
|---|
| AID1455145 | Inhibition of recombinant human MAGL expressed in African green monkey COS7 cells using 2-arachidonoyl-[3H]-glycerol as substrate after 20 mins by scintillation counting analysis | 2018 | Journal of medicinal chemistry, 02-08, Volume: 61, Issue:3
| Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors. |
| AID389888 | Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cells by scintillation counting | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389889 | Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells by scintillation counting | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID362906 | Inhibition of human recombinant fatty acid synthase thioesterase domain by fluorogenic assay | 2008 | Journal of medicinal chemistry, Sep-11, Volume: 51, Issue:17
| Synthesis of novel beta-lactone inhibitors of fatty acid synthase. |
| AID389886 | Inhibition of human recombinant DAGL-alpha-mediated sn-1-[14C]oleoyl-2-arachidonoyl-glycerol hydrolysis to 2-AG overexpressed in african green monkey COS7 cell membrane by scintillation counting | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389895 | Selectivity ratio of IC50 for african green monkey MAGL over IC50 for human recombinant DAGLalpha | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389890 | Inhibition of FAAH-mediated [14C]anandamide hydrolysis in rat brain membrane | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID362903 | Cytotoxicity against human Hs 58.Fs cells after 48 hrs by Cell titer assay | 2008 | Journal of medicinal chemistry, Sep-11, Volume: 51, Issue:17
| Synthesis of novel beta-lactone inhibitors of fatty acid synthase. |
| AID1185868 | Inhibition of MGL in African green monkey COS7 cells cytosolic fraction assessed as reduction in 2-arachidonoyl-[3H]-glycerol hydrolysis at 1 uM by scintillation counting method | 2014 | Bioorganic & medicinal chemistry, Sep-01, Volume: 22, Issue:17
| Structure-affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist. |
| AID389887 | Inhibition of MAGL-mediated [14C]2-arachidonoyl glycerol hydrolysis to [3H]arachidonic acid in african green monkey COS cell cytosolic fraction by scintillation counting | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389897 | Selectivity ratio of IC50 for african green monkey MAGL over Ki for human recombinant CB2 receptor | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389898 | Selectivity ratio of IC50 for african green monkey MAGL over IC50 for rat brain membrane FAAH | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID389900 | Enhancement of ionomycin-induced stimulation of 2-AG biosynthesis in mouse N18TG2 cells at 1.5 uM | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID362907 | Ratio of IC50 for human Hs 58.Fs cells to IC50 for human MDA-MB-435 cells | 2008 | Journal of medicinal chemistry, Sep-11, Volume: 51, Issue:17
| Synthesis of novel beta-lactone inhibitors of fatty acid synthase. |
| AID362905 | Cytotoxicity against human MDA-MB-435 cells after 48 hrs by Cell titer assay | 2008 | Journal of medicinal chemistry, Sep-11, Volume: 51, Issue:17
| Synthesis of novel beta-lactone inhibitors of fatty acid synthase. |
| AID389896 | Selectivity ratio of IC50 for african green monkey MAGL over Ki for human recombinant CB1 receptor | 2008 | Journal of medicinal chemistry, Nov-13, Volume: 51, Issue:21
| Tetrahydrolipstatin analogues as modulators of endocannabinoid 2-arachidonoylglycerol metabolism. |
| AID1798446 | Fluorogenic Assay for Detection of FASTE Inhibition from Article 10.1021/jm800321h: \\Synthesis of novel beta-lactone inhibitors of fatty acid synthase.\\ | 2008 | Journal of medicinal chemistry, Sep-11, Volume: 51, Issue:17
| Synthesis of novel beta-lactone inhibitors of fatty acid synthase. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |