Assay ID | Title | Year | Journal | Article |
AID1211541 | Drug metabolism in human urine assessed as (1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211519 | Drug metabolism assessed as human recombinant CYP2E1-mediated (1-(5-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211522 | Drug metabolism assessed as human recombinant CYP3A4-mediated (1-(5-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211526 | Drug metabolism assessed as human recombinant CYP3A4-mediated (1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211525 | Drug metabolism assessed as human recombinant CYP2E1-mediated (1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211520 | Drug metabolism assessed as human recombinant CYP2E1-mediated 5-(3-(1-naphthoyl)-1H-indol-1-yl)pentanoic acid formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211515 | Activation of CB1 receptor in B6SJL mouse brain membrane assessed as [35S]-GTPgammaS binding at 10 uM after 30 mins by liquid scintillation spectrophotometric analysis in presence of O-2050 | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211523 | Drug metabolism assessed as human recombinant CYP3A4-mediated 5-(3-(1-naphthoyl)-1H-indol-1-yl)pentanoic acid formation at 10 uM after 90 mins by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211513 | Displacement of [3H]CP-55,940 from CB1 receptor in B6SJL mouse brain membrane after 90 mins by liquid scintillation spectrophotometric analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211514 | Activation of CB1 receptor in B6SJL mouse brain membrane assessed as [35S]-GTPgammaS binding at 10 uM after 30 mins by liquid scintillation spectrophotometric analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211539 | Drug metabolism in human urine assessed as 5-(3-(1-naphthoyl)-1H-indol-1-yl)pentanoic acid formation by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1211540 | Drug metabolism in human urine assessed as (1-(5-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone formation by LC-MS/MS analysis | 2012 | Drug metabolism and disposition: the biological fate of chemicals, Nov, Volume: 40, Issue:11
| Cytochrome P450-mediated oxidative metabolism of abused synthetic cannabinoids found in K2/Spice: identification of novel cannabinoid receptor ligands. |
AID1346701 | Human CB1 receptor (Cannabinoid receptors) | 2015 | ACS chemical neuroscience, Aug-19, Volume: 6, Issue:8
| Effects of bioisosteric fluorine in synthetic cannabinoid designer drugs JWH-018, AM-2201, UR-144, XLR-11, PB-22, 5F-PB-22, APICA, and STS-135. |
AID1346728 | Human CB2 receptor (Cannabinoid receptors) | 2015 | ACS chemical neuroscience, Aug-19, Volume: 6, Issue:8
| Effects of bioisosteric fluorine in synthetic cannabinoid designer drugs JWH-018, AM-2201, UR-144, XLR-11, PB-22, 5F-PB-22, APICA, and STS-135. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |