| 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 | Bos taurus (cattle) | IC50 | 29.0000 | 1 | 1 |
| 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 | Homo sapiens (human) | IC50 | 29.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Sus scrofa (pig) | Ki | 4.0940 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 2.5550 | 1 | 1 |
| 72 kDa type IV collagenase | Homo sapiens (human) | IC50 | 30.3100 | 1 | 1 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 4.8000 | 1 | 1 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 1.5400 | 1 | 1 |
| calpain II, partial | Sus scrofa (pig) | IC50 | 1.7742 | 1 | 1 |
| Calpain-1 catalytic subunit | Homo sapiens (human) | IC50 | 23.4200 | 3 | 3 |
| Calpain-1 catalytic subunit | Sus scrofa (pig) | IC50 | 0.0800 | 1 | 1 |
| Cannabinoid receptor 2 | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| Cathepsin B | Bos taurus (cattle) | IC50 | 0.3100 | 1 | 1 |
| Cathepsin B | Homo sapiens (human) | IC50 | 4.8155 | 3 | 3 |
| Cathepsin B | Homo sapiens (human) | Ki | 0.0063 | 3 | 3 |
| Cathepsin B | Capra hircus (goat) | Ki | 0.0063 | 2 | 2 |
| Cathepsin G | Homo sapiens (human) | IC50 | 1.1000 | 1 | 1 |
| Cathepsin G | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| Cathepsin K | Homo sapiens (human) | Ki | 0.0240 | 1 | 1 |
| Cationic trypsin | Bos taurus (cattle) | IC50 | 8.1000 | 1 | 1 |
| Cysteine protease | Leishmania donovani | IC50 | 0.0100 | 1 | 1 |
| Cysteine protease falcipain-3 | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0925 | 2 | 2 |
| Cysteine proteinase falcipain 2a | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0636 | 3 | 3 |
| Cytosolic phospholipase A2 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 1.2410 | 1 | 1 |
| Delta-type opioid receptor | Homo sapiens (human) | Ki | 0.0362 | 2 | 2 |
| Delta-type opioid receptor | Sus scrofa (pig) | Ki | 0.0365 | 1 | 1 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit delta | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit pi | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit theta | Homo sapiens (human) | Ki | 0.0060 | 2 | 2 |
| Group 10 secretory phospholipase A2 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Hepatocyte growth factor activator | Homo sapiens (human) | Ki | 0.1880 | 1 | 1 |
| hypothetical protein SA1422 | Staphylococcus aureus subsp. aureus N315 | IC50 | 19.3900 | 2 | 2 |
| M1-family alanyl aminopeptidase | Plasmodium falciparum 3D7 | IC50 | 108.3900 | 1 | 1 |
| Matrix metalloproteinase-9 | Homo sapiens (human) | IC50 | 2.5800 | 1 | 1 |
| Mcl-1 | Homo sapiens (human) | IC50 | 1.6341 | 1 | 1 |
| Myeloblastin | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 1.2700 | 1 | 1 |
| Neutrophil elastase | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| Papain | Carica papaya (papaya) | IC50 | 0.0022 | 1 | 1 |
| Papain | Carica papaya (papaya) | Ki | 52.0000 | 1 | 1 |
| Phospholipase A2 | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Phospholipase A2, membrane associated | Homo sapiens (human) | IC50 | 23.8000 | 1 | 1 |
| Plasma kallikrein | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Plasminogen | Homo sapiens (human) | IC50 | 1.2000 | 1 | 1 |
| Plasminogen | Bos taurus (cattle) | IC50 | 3.7000 | 1 | 1 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | IC50 | 0.1023 | 3 | 3 |
| Poly [ADP-ribose] polymerase 2 | Homo sapiens (human) | IC50 | 10.3000 | 2 | 2 |
| Pro-cathepsin H | Homo sapiens (human) | Ki | 9.2000 | 2 | 2 |
| Procathepsin L | Homo sapiens (human) | IC50 | 2.6798 | 4 | 4 |
| Prothrombin | Bos taurus (cattle) | IC50 | 12.0000 | 1 | 1 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | IC50 | 8.3000 | 1 | 1 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 8.3000 | 1 | 1 |
| Replicase polyprotein 1ab | Human coronavirus 229E | IC50 | 8.3000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 8.3000 | 2 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 8.3000 | 3 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Ki | 13.8000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | Ki | 13.8000 | 2 | 2 |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | IC50 | 119.0000 | 1 | 1 |
| Serine protease hepsin | Homo sapiens (human) | Ki | 0.0610 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | IC50 | 8.3000 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | IC50 | 8.3000 | 1 | 1 |
| Stromelysin-1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Suppressor of tumorigenicity 14 protein | Homo sapiens (human) | Ki | 1.2980 | 2 | 2 |
| Transmembrane protease serine 2 | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| Transmembrane protease serine 6 | Homo sapiens (human) | Ki | 3.2500 | 2 | 2 |
| Trypsin | Sus scrofa (pig) | IC50 | 0.3500 | 2 | 2 |
| Trypsin-1 | Homo sapiens (human) | IC50 | 0.6000 | 1 | 1 |
| Trypsin-2 | Homo sapiens (human) | IC50 | 0.6000 | 1 | 1 |
| Trypsin-3 | Homo sapiens (human) | IC50 | 0.6000 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 7.4000 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | Ki | 7.8000 | 1 | 1 |
| Valosin-containing protein | Homo sapiens (human) | IC50 | 36.3280 | 2 | 3 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | IC50 | 35.3000 | 1 | 1 |