A calpain-1 catalytic subunit that is encoded in the genome of pig. [OMA:P35750, PRO:DNx]
EC 3.4.22.52;
Calcium-activated neutral proteinase 1;
CANP 1;
Calpain mu-type;
Calpain-1 large subunit;
Micromolar-calpain;
muCANP
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 5 (55.56) | 29.6817 |
| 2010's | 3 (33.33) | 24.3611 |
| 2020's | 1 (11.11) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| leupeptin | Sus scrofa (pig) | IC50 | 0.0800 | 1 | 1 |
| carbobenzoxyvalylphenylalanine aldehyde | Sus scrofa (pig) | Ki | 0.0100 | 1 | 1 |
| e 64 | Sus scrofa (pig) | Ki | 3.9600 | 1 | 1 |
| ak 295 | Sus scrofa (pig) | Ki | 0.1500 | 1 | 1 |
| acetylleucyl-leucyl-norleucinal | Sus scrofa (pig) | Ki | 0.1900 | 1 | 1 |
| pd 150606 | Sus scrofa (pig) | IC50 | 18.5500 | 2 | 2 |
| sja 6017 | Sus scrofa (pig) | IC50 | 0.0213 | 2 | 2 |
| calpain inhibitor iii | Sus scrofa (pig) | IC50 | 0.0200 | 1 | 1 |
| calpain inhibitor iii | Sus scrofa (pig) | Ki | 0.0100 | 1 | 1 |
| amg 853 | Sus scrofa (pig) | IC50 | 53.7500 | 2 | 2 |