Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 25.6651 | 1 | 2 |
15-lipoxygenase, partial | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
67.9K protein | Vaccinia virus | Potency | 9.3146 | 2 | 8 |
acetylcholinesterase | Homo sapiens (human) | Potency | 34.1947 | 3 | 6 |
aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 14.4728 | 1 | 3 |
alpha-galactosidase | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
AR protein | Homo sapiens (human) | Potency | 14.1170 | 10 | 22 |
aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 22.4240 | 2 | 6 |
Ataxin-2 | Homo sapiens (human) | Potency | 20.1469 | 1 | 3 |
ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 18.7094 | 2 | 4 |
Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 23.1837 | 2 | 5 |
caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 4.8620 | 1 | 4 |
Caspase-7 | Homo sapiens (human) | Potency | 3.9946 | 1 | 3 |
Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 6.1071 | 3 | 7 |
cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 3.0016 | 2 | 3 |
Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 2.2247 | 1 | 3 |
Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 28.4514 | 1 | 4 |
Chain A, Breast cancer type 1 susceptibility protein | Homo sapiens (human) | Potency | 18.4029 | 2 | 4 |
Chain A, Cruzipain | Trypanosoma cruzi | Potency | 25.1189 | 1 | 1 |
Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 31.6228 | 1 | 1 |
Chain A, HADH2 protein | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 64.7758 | 1 | 2 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 21.1789 | 2 | 5 |
Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 1.3511 | 1 | 3 |
Chain B, HADH2 protein | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
chromobox protein homolog 1 | Homo sapiens (human) | Potency | 59.9574 | 1 | 3 |
core-binding factor subunit beta isoform 2 | Homo sapiens (human) | Potency | 6.9603 | 3 | 5 |
cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 1.5849 | 1 | 1 |
cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 27.5404 | 1 | 1 |
cytochrome P450 2D6 | Homo sapiens (human) | Potency | 3.4671 | 1 | 1 |
cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 6.3096 | 1 | 1 |
cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 14.3194 | 2 | 8 |
cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 1.5487 | 1 | 1 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 19.1907 | 1 | 3 |
Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | Potency | 0.6310 | 1 | 1 |
DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 35.4668 | 2 | 6 |
DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 14.3412 | 2 | 7 |
DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 14.4126 | 2 | 14 |
estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 28.1831 | 10 | 20 |
estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 9.9008 | 1 | 2 |
estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 5.3824 | 6 | 12 |
euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 12.1508 | 1 | 4 |
farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 8.9317 | 3 | 5 |
flap endonuclease 1 | Homo sapiens (human) | Potency | 10.8395 | 2 | 5 |
Fumarate hydratase | Homo sapiens (human) | Potency | 4.4668 | 1 | 1 |
G | Vesicular stomatitis virus | Potency | 27.5404 | 1 | 1 |
GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 14.3194 | 1 | 4 |
geminin | Homo sapiens (human) | Potency | 13.6838 | 2 | 6 |
GLI family zinc finger 3 | Homo sapiens (human) | Potency | 22.6716 | 2 | 4 |
glp-1 receptor, partial | Homo sapiens (human) | Potency | 3.7298 | 1 | 3 |
glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 5.5035 | 3 | 5 |
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | Potency | 6.3096 | 1 | 1 |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 18.2028 | 2 | 3 |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | Potency | 6.3096 | 1 | 1 |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | Potency | 6.3096 | 1 | 1 |
GTP-binding nuclear protein Ran isoform 1 | Homo sapiens (human) | Potency | 0.2372 | 1 | 2 |
Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 29.5947 | 1 | 3 |
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 27.7170 | 1 | 2 |
heat shock protein beta-1 | Homo sapiens (human) | Potency | 25.0654 | 1 | 2 |
hemoglobin subunit beta | Homo sapiens (human) | Potency | 2.5119 | 2 | 2 |
Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 12.5893 | 1 | 3 |
histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 19.4549 | 1 | 4 |
Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 80.0112 | 2 | 2 |
histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 41.1572 | 1 | 4 |
HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 27.5404 | 1 | 1 |
huntingtin isoform 2 | Homo sapiens (human) | Potency | 14.7755 | 1 | 4 |
hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 26.0297 | 2 | 3 |
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
IDH1 | Homo sapiens (human) | Potency | 7.3551 | 1 | 3 |
importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 0.2372 | 1 | 2 |
Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 27.5404 | 1 | 2 |
Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 19.7020 | 1 | 2 |
Integrin alpha-IIb | Homo sapiens (human) | Potency | 3.9811 | 1 | 1 |
Integrin beta-3 | Homo sapiens (human) | Potency | 3.9811 | 1 | 1 |
Interferon beta | Homo sapiens (human) | Potency | 27.5404 | 1 | 1 |
lamin isoform A-delta10 | Homo sapiens (human) | Potency | 17.5864 | 1 | 3 |
lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 2.5119 | 1 | 1 |
luciferase | Photuris pensylvanica (Pennsylania firefly) | Potency | 15.8489 | 1 | 1 |
Microtubule-associated protein tau | Homo sapiens (human) | Potency | 5.3440 | 2 | 7 |
mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 9.5325 | 3 | 4 |
nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 5.0001 | 2 | 5 |
nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 18.4675 | 1 | 2 |
nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 16.7487 | 2 | 10 |
nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 17.9584 | 2 | 4 |
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 75.6863 | 1 | 1 |
peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 7.1313 | 2 | 4 |
peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 40.0648 | 3 | 4 |
peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 26.5881 | 2 | 3 |
phosphopantetheinyl transferase | Bacillus subtilis | Potency | 40.9903 | 1 | 3 |
plasminogen precursor | Mus musculus (house mouse) | Potency | 1.1904 | 1 | 2 |
Platelet-activating factor receptor | Homo sapiens (human) | Potency | 29.8816 | 1 | 2 |
polyprotein | Zika virus | Potency | 4.4668 | 1 | 1 |
progesterone receptor | Homo sapiens (human) | Potency | 25.8539 | 1 | 2 |
Rap guanine nucleotide exchange factor 3 | Homo sapiens (human) | Potency | 46.8078 | 2 | 4 |
Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 75.4550 | 2 | 4 |
retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 23.3010 | 3 | 6 |
retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 4.5186 | 3 | 3 |
runt-related transcription factor 1 isoform AML1b | Homo sapiens (human) | Potency | 6.9603 | 3 | 5 |
serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 0.5030 | 1 | 2 |
Smad3 | Homo sapiens (human) | Potency | 6.5655 | 1 | 4 |
snurportin-1 | Homo sapiens (human) | Potency | 0.2372 | 1 | 2 |
survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 10.0000 | 1 | 2 |
TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
TDP1 protein | Homo sapiens (human) | Potency | 1.2177 | 2 | 14 |
thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 25.7084 | 2 | 6 |
thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 33.2482 | 4 | 10 |
thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 31.1402 | 6 | 10 |
transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 30.3803 | 1 | 3 |
tumor necrosis factor | Homo sapiens (human) | Potency | 37.5780 | 1 | 1 |
tumor susceptibility gene 101 protein | Homo sapiens (human) | Potency | 10.0000 | 1 | 2 |
ubiquitin carboxyl-terminal hydrolase 2 isoform a | Homo sapiens (human) | Potency | 0.6310 | 1 | 1 |
urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 1.1904 | 1 | 2 |
urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 1.1904 | 1 | 2 |
USP1 protein, partial | Homo sapiens (human) | Potency | 21.7984 | 2 | 6 |
v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 21.7761 | 1 | 1 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 15.6968 | 1 | 2 |
vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 30.7089 | 1 | 7 |
Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 24.1495 | 1 | 2 |
Vpr | Human immunodeficiency virus 1 | Potency | 9.0532 | 1 | 2 |
WRN | Homo sapiens (human) | Potency | 13.3188 | 2 | 5 |