Page last updated: 2024-08-07 22:56:10

insulin-degrading enzyme isoform 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (24)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
2-[[[5-(3-chlorophenyl)-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-1H-benzimidazoleHomo sapiens (human)IC502.974740
N-[(tert-butylamino)-oxomethyl]-2-[4-(3-chlorophenyl)-1-piperazinyl]acetamideHomo sapiens (human)IC5055.941010
2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-oneHomo sapiens (human)IC504.054010
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidHomo sapiens (human)IC502.102010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
acriflavine chlorideHomo sapiens (human)EC5054.727020
pyronineHomo sapiens (human)EC5054.732020
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineHomo sapiens (human)EC5054.686020
topotecan hydrochlorideHomo sapiens (human)EC5054.690020
daunorubicin hydrochlorideHomo sapiens (human)EC5054.705020
diacetylfluoresceinHomo sapiens (human)EC5054.710020
habaHomo sapiens (human)EC5024.583520
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dioneHomo sapiens (human)EC5054.661020
pd 147953Homo sapiens (human)EC5014.556020
biotinHomo sapiens (human)EC502.449520
brazilinHomo sapiens (human)EC5054.669020
desthiobiotinHomo sapiens (human)EC507.601520
calmidazoliumHomo sapiens (human)EC5028.368020
2-(4-bromophenoxy)-N-[(2-hydroxy-5-methylanilino)-sulfanylidenemethyl]acetamideHomo sapiens (human)EC5054.691020
N-[2-(4-methoxyphenoxy)ethyl]-5-(4-morpholinyl)-2-nitroanilineHomo sapiens (human)EC5054.732020
6-phenylspiro[7-oxa-1-azabicyclo[2.2.1]heptane-2,1'-cyclopentane]Homo sapiens (human)EC5054.692020
n-oleoyldopamineHomo sapiens (human)EC5031.824020
2-(2-furanylmethyl)-3-[[2-(3-pyridinyl)-3H-benzimidazol-5-yl]amino]-3H-isoindol-1-oneHomo sapiens (human)EC5054.646020
3,6-diamino-10-methylacridinium chloride hydrochlorideHomo sapiens (human)EC5054.721020
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)EC5034.524520