Assay ID | Title | Year | Journal | Article |
AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1139350 | Inhibition of delta opioid receptor (unknown origin) using SNC-80 by high content imaging beta-arrestin translocation assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139357 | Binding affinity to NET (unknown origin) | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1859165 | Antagonist at KOR expressed in human U2OS cells measured by High content imaging based beta-arrestin translocation assay | 2022 | European journal of medicinal chemistry, Feb-05, Volume: 229 | Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities. |
AID1139352 | Binding affinity to histamine H1 receptor (unknown origin) | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139362 | Selectivity ratio of IC50 for delta opioid receptor (unknown origin) by HCS assay to IC50 for kappa opioid receptor (unknown origin) by DRx assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139347 | Inhibition of mu opioid receptor (unknown origin) using DAMGO by high content imaging beta-arrestin translocation assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139359 | Binding affinity to dopamine D3 receptor (unknown origin) | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139364 | Drug metabolism in mouse liver microsomes assessed as compound remaining after 1 hr | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139361 | Selectivity ratio of IC50 for mu opioid receptor (unknown origin) by HCS assay to IC50 for kappa opioid receptor (unknown origin) by DRx assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1139348 | Inhibition of kappa opioid receptor (unknown origin) using dynorphin A by DiscoveryRx b-arrestin PathHunter assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
AID1859167 | Metabolic stability in human liver microsomes assessed as compound remaining after 1 hr | 2022 | European journal of medicinal chemistry, Feb-05, Volume: 229 | Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities. |
AID1859166 | Permeability of the compound across blood brain barrier at pH 7.4 by PAMPA | 2022 | European journal of medicinal chemistry, Feb-05, Volume: 229 | Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activities. |
AID1139349 | Inhibition of kappa opioid receptor (unknown origin) using dynorphin A by high content imaging beta-arrestin translocation assay | 2014 | Bioorganic & medicinal chemistry letters, May-01, Volume: 24, Issue:9
| Antagonists of the kappa opioid receptor. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |