| Assay ID | Title | Year | Journal | Article |
|---|
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1069374 | Antiproliferative activity against human MIAPaCa2 cells after 96 hrs by CyQuant-based assay in presence of NMN | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069380 | Antiproliferative activity against human HT1080 cells after 96 hrs by CyQuant-based assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069383 | Antiproliferative activity against human A2780 cells after 72 hrs by SRB assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1064301 | Cytotoxicity against human RCC4/VHL cells after 4 days by XTT assay | 2014 | Bioorganic & medicinal chemistry, Jan-15, Volume: 22, Issue:2
| Identifying novel targets in renal cell carcinoma: design and synthesis of affinity chromatography reagents. |
| AID1069375 | Antiproliferative activity against human HT1080 cells after 96 hrs by CyQuant-based assay in presence of NMN | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069385 | Inhibition of full length C-terminal His6-tagged human NAMPT expressed in Escherichia coli Rosetta (DE3) cells using PRPP/NAM as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measured after 30 mins | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1425907 | Growth inhibition of VHL-deficient human RCC4 cells by XTT assay | 2016 | MedChemComm, Sep-01, Volume: 7, Issue:9
| Anticancer agents interacting with membrane glucose transporters. |
| AID1064300 | Selectivity ratio of IC50 for human RCC4/VHL cells to IC50 for human RCC4 cells | 2014 | Bioorganic & medicinal chemistry, Jan-15, Volume: 22, Issue:2
| Identifying novel targets in renal cell carcinoma: design and synthesis of affinity chromatography reagents. |
| AID1069379 | Antiproliferative activity against human PC3 cells after 96 hrs by CyQuant-based assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069373 | Antiproliferative activity against human HCT116 cells after 96 hrs by CyQuant-based assay in presence of NMN | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069377 | Antiproliferative activity against human HCT116 cells after 96 hrs by CyQuant-based assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069381 | Inhibition of NAMPT in human A2780 cells assessed as reduction in NAD level after 48 hrs by LC-MS/MS analysis | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069378 | Antiproliferative activity against human MIAPaCa2 cells after 96 hrs by CyQuant-based assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1069376 | Antiproliferative activity against human PC3 cells after 96 hrs by CyQuant-based assay in presence of NMN | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| AID1064302 | Cytotoxicity against human RCC4 cells after 4 days by XTT assay | 2014 | Bioorganic & medicinal chemistry, Jan-15, Volume: 22, Issue:2
| Identifying novel targets in renal cell carcinoma: design and synthesis of affinity chromatography reagents. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | 2014 | Journal of biomolecular screening, Jul, Volume: 19, Issue:6
| A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | | | |
| AID977608 | Experimentally measured binding affinity data (IC50) for protein-ligand complexes derived from PDB | 2014 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 24, Issue:3
| Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT). |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |