| Assay ID | Title | Year | Journal | Article |
|---|
| AID740005 | Hypothermic effect in Sprague-Dawley rat assessed as decrease in core body temperature at 10 mg/kg | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID238865 | Inhibition of [3H]CP-55940 binding to cannabinoid receptor 1 of rat brain | 2005 | Journal of medicinal chemistry, Jul-14, Volume: 48, Issue:14
| Adamantyl cannabinoids: a novel class of cannabinergic ligands. |
| AID262341 | Displacement of [3H]CP-55940 from mouse spleen CB2 receptor | 2006 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 16, Issue:6
| Structural modifications of the cannabinoid side chain towards C3-aryl and 1',1'-cycloalkyl-1'-cyano cannabinoids. |
| AID740014 | Selectivity ratio of Ki for mouse CB2 receptor to Ki for rat CB1 receptor | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID740008 | Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 mins relative to WIN55,212-2 | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID247066 | In vivo cannabinergic activity in rat after 90 min of dose administration (0.03-1.8 mg/kg) using drug discrimination assay | 2005 | Journal of medicinal chemistry, Jul-14, Volume: 48, Issue:14
| Adamantyl cannabinoids: a novel class of cannabinergic ligands. |
| AID416356 | Binding affinity to CB2 receptor | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Quantitative structure-activity relationship (QSAR) for a series of novel cannabinoid derivatives using descriptors derived from semi-empirical quantum-chemical calculations. |
| AID740003 | Antinociceptive activity in Sprague-Dawley rat assessed as increase in tail-flick latency period at 0.05 mg/kg, sc by tail-flick test | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID311038 | Binding affinity to CB2 receptor | 2007 | Journal of medicinal chemistry, Jun-14, Volume: 50, Issue:12
| The application of 3D-QSAR studies for novel cannabinoid ligands substituted at the C1' position of the alkyl side chain on the structural requirements for binding to cannabinoid receptors CB1 and CB2. |
| AID262340 | Displacement of [3H]CP-55940 from rat brain CB1 receptor | 2006 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 16, Issue:6
| Structural modifications of the cannabinoid side chain towards C3-aryl and 1',1'-cycloalkyl-1'-cyano cannabinoids. |
| AID740016 | Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in mouse spleen membrane by competitive binding assay | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID391587 | Displacement of [3H]CP-55940 from CB2 receptor in mouse spleen membrane | 2008 | Journal of medicinal chemistry, Oct-23, Volume: 51, Issue:20
| Bornyl- and isobornyl-Delta8-tetrahydrocannabinols: a novel class of cannabinergic ligands. |
| AID416355 | Binding affinity to CB1 receptor | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Quantitative structure-activity relationship (QSAR) for a series of novel cannabinoid derivatives using descriptors derived from semi-empirical quantum-chemical calculations. |
| AID740002 | Antinociceptive activity in Sprague-Dawley rat assessed as increase in tail-flick latency period at 0.1 to 10 mg/kg, sc after 60 to 120 mins by tail-flick test | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID391586 | Displacement of [3H]CP-55940 from CB1 receptor in rat brain synaptosome membrane | 2008 | Journal of medicinal chemistry, Oct-23, Volume: 51, Issue:20
| Bornyl- and isobornyl-Delta8-tetrahydrocannabinols: a novel class of cannabinergic ligands. |
| AID247069 | In vivo cannabinergic activity in rat after 30 min of dose administration (0.03-1.8 mg/kg) using drug discrimination assay | 2005 | Journal of medicinal chemistry, Jul-14, Volume: 48, Issue:14
| Adamantyl cannabinoids: a novel class of cannabinergic ligands. |
| AID262342 | Selectivity for rat CB1 receptor over mouse CB2 receptor | 2006 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 16, Issue:6
| Structural modifications of the cannabinoid side chain towards C3-aryl and 1',1'-cycloalkyl-1'-cyano cannabinoids. |
| AID496926 | Displacement of [3H]CP-55940 from CB1 receptor in rat brain | 2010 | Journal of medicinal chemistry, Aug-12, Volume: 53, Issue:15
| Heteroadamantyl cannabinoids. |
| AID311037 | Binding affinity to CB1 receptor | 2007 | Journal of medicinal chemistry, Jun-14, Volume: 50, Issue:12
| The application of 3D-QSAR studies for novel cannabinoid ligands substituted at the C1' position of the alkyl side chain on the structural requirements for binding to cannabinoid receptors CB1 and CB2. |
| AID740007 | Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 mins | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID569313 | Displacement of [3H]CP 55940 from human CB2 receptor in cell free system | 2011 | European journal of medicinal chemistry, Feb, Volume: 46, Issue:2
| Three-dimensional quantitative structure-selectivity relationships analysis guided rational design of a highly selective ligand for the cannabinoid receptor 2. |
| AID496928 | Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cell membranes | 2010 | Journal of medicinal chemistry, Aug-12, Volume: 53, Issue:15
| Heteroadamantyl cannabinoids. |
| AID496927 | Displacement of [3H]CP-55940 from mouse CB2 receptor expressed in HEK293 cell membranes | 2010 | Journal of medicinal chemistry, Aug-12, Volume: 53, Issue:15
| Heteroadamantyl cannabinoids. |
| AID239117 | Inhibition of [3H]CP-55940 binding to cannabinoid receptor 2 of mouse spleen membranes | 2005 | Journal of medicinal chemistry, Jul-14, Volume: 48, Issue:14
| Adamantyl cannabinoids: a novel class of cannabinergic ligands. |
| AID740017 | Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assay | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| AID740001 | Antinociceptive activity in Sprague-Dawley rat assessed as increase in tail-flick latency period at 0.1 to 10 mg/kg, sc after 6 hrs by tail-flick test | 2013 | Journal of medicinal chemistry, May-23, Volume: 56, Issue:10
| Novel adamantyl cannabinoids as CB1 receptor probes. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |