| Assay ID | Title | Year | Journal | Article |
|---|
| AID416355 | Binding affinity to CB1 receptor | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Quantitative structure-activity relationship (QSAR) for a series of novel cannabinoid derivatives using descriptors derived from semi-empirical quantum-chemical calculations. |
| AID49845 | Binding affinity towards Cannabinoid receptor 2 using CP-55940 as radioligand in HEK293 EBNA cells | 2003 | Bioorganic & medicinal chemistry letters, Oct-20, Volume: 13, Issue:20
| Synthesis and testing of novel phenyl substituted side-chain analogues of classical cannabinoids. |
| AID311038 | Binding affinity to CB2 receptor | 2007 | Journal of medicinal chemistry, Jun-14, Volume: 50, Issue:12
| The application of 3D-QSAR studies for novel cannabinoid ligands substituted at the C1' position of the alkyl side chain on the structural requirements for binding to cannabinoid receptors CB1 and CB2. |
| AID416356 | Binding affinity to CB2 receptor | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Quantitative structure-activity relationship (QSAR) for a series of novel cannabinoid derivatives using descriptors derived from semi-empirical quantum-chemical calculations. |
| AID414287 | Binding affinity to human CB2 receptor transfected in HEK293 cells | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Design and synthesis of novel tri-aryl CB2 selective cannabinoid ligands. |
| AID49314 | Binding affinity towards Cannabinoid receptor 1 using CP-55940 as radioligand in HEK293 EBNA cells | 2003 | Bioorganic & medicinal chemistry letters, Oct-20, Volume: 13, Issue:20
| Synthesis and testing of novel phenyl substituted side-chain analogues of classical cannabinoids. |
| AID414286 | Binding affinity to human CB1 receptor transfected in HEK293 cells | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Design and synthesis of novel tri-aryl CB2 selective cannabinoid ligands. |
| AID406568 | Cytotoxicity against human DBTRG-O5MG cells assessed as cell death after 18 hrs | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID406564 | Cytotoxicity against human U87 cells by side flank model relative to control | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID311037 | Binding affinity to CB1 receptor | 2007 | Journal of medicinal chemistry, Jun-14, Volume: 50, Issue:12
| The application of 3D-QSAR studies for novel cannabinoid ligands substituted at the C1' position of the alkyl side chain on the structural requirements for binding to cannabinoid receptors CB1 and CB2. |
| AID406561 | Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cells | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID49327 | Ratio of binding affinity towards cannabinoid receptor-1 (CB1) to that of cannabinoid receptor-2 (CB2) | 2003 | Bioorganic & medicinal chemistry letters, Oct-20, Volume: 13, Issue:20
| Synthesis and testing of novel phenyl substituted side-chain analogues of classical cannabinoids. |
| AID406569 | Cytotoxicity against human MT310 cells assessed as cell death after 18 hrs | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID414288 | Selectivity ratio of Ki for human CB1 receptor to Ki for human CB2 receptor | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Design and synthesis of novel tri-aryl CB2 selective cannabinoid ligands. |
| AID406565 | Cytotoxicity against human U87MG cells assessed as cell death after 18 hrs | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID406567 | Cytotoxicity against human LN229 cells assessed as cell death after 18 hrs | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID406566 | Cytotoxicity against human T98G cells assessed as cell death after 18 hrs | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID406562 | Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cells | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| AID406563 | Selectivity ratio of Ki for human CB1 receptor to Ki for human CB2 receptor | 2008 | Bioorganic & medicinal chemistry, Jul-01, Volume: 16, Issue:13
| Exploring the substituent effects on a novel series of C1'-dimethyl-aryl Delta8-tetrahydrocannabinol analogs. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |