| Assay ID | Title | Year | Journal | Article |
|---|
| AID208984 | Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucrase | 1986 | Journal of medicinal chemistry, Jun, Volume: 29, Issue:6
| Synthesis and alpha-D-glucosidase inhibitory activity of N-substituted valiolamine derivatives as potential oral antidiabetic agents. |
| AID104666 | Inhibitory activity against porcine maltase | 1986 | Journal of medicinal chemistry, Jun, Volume: 29, Issue:6
| Synthesis and alpha-D-glucosidase inhibitory activity of N-substituted valiolamine derivatives as potential oral antidiabetic agents. |
| AID342793 | Inhibition of rat intestinal brush border membrane maltase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID1895992 | Inhibition of full length human recombinant Endoplasmic reticulum alpha-glucosidase 1 expressed in Escherichia coli using trisaccharide as substrate incubated for 60 mins | 2021 | Journal of medicinal chemistry, 12-23, Volume: 64, Issue:24
| N-Substituted Valiolamine Derivatives as Potent Inhibitors of Endoplasmic Reticulum α-Glucosidases I and II with Antiviral Activity. |
| AID342795 | Inhibition of rat intestinal brush border membrane isomaltase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID342804 | Inhibition of rabbit glycogen phosphorylase B at 400 uM | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID1895996 | Antiviral activity against SARS-CoV-2 England/2/2022 assessed as reduction in viral infection | 2021 | Journal of medicinal chemistry, 12-23, Volume: 64, Issue:24
| N-Substituted Valiolamine Derivatives as Potent Inhibitors of Endoplasmic Reticulum α-Glucosidases I and II with Antiviral Activity. |
| AID342805 | Inhibition of rabbit muscle amylo-1,6-glucosidase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID342797 | Inhibition of rat intestinal brush border membrane sucrase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID342802 | Inhibition of human lysosomal beta-glucosidase at 1000 uM | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID1895994 | Cytotoxicity against African green monkey Vero cells assessed as reduction in cell viability incubated for 3 to 5 days by Cell titer-glo luminescent assay | 2021 | Journal of medicinal chemistry, 12-23, Volume: 64, Issue:24
| N-Substituted Valiolamine Derivatives as Potent Inhibitors of Endoplasmic Reticulum α-Glucosidases I and II with Antiviral Activity. |
| AID342809 | Inhibition of pig intestinal maltase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID342810 | Inhibition of pig intestinal sucrase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID342799 | Inhibition of human lysosomal alpha-glucosidase | 2008 | Bioorganic & medicinal chemistry, Aug-01, Volume: 16, Issue:15
| In vitro inhibition of glycogen-degrading enzymes and glycosidases by six-membered sugar mimics and their evaluation in cell cultures. |
| AID1895993 | Inhibition of full length N-terminal his6-tagged mouse recombinant Endoplasmic reticulum alpha-glucosidase 2 expressed in DH10 Escherichia coli using Fluorogenic 1,4-methyl-lumbelliferon as substrate preincubated for 60 mins followed by substrate addition | 2021 | Journal of medicinal chemistry, 12-23, Volume: 64, Issue:24
| N-Substituted Valiolamine Derivatives as Potent Inhibitors of Endoplasmic Reticulum α-Glucosidases I and II with Antiviral Activity. |
| AID1895995 | Antiviral activity against DENV New Guinea C strain infected in African green monkey Vero cells assessed as reduction in viral infection measured after 5 days by plaque assay | 2021 | Journal of medicinal chemistry, 12-23, Volume: 64, Issue:24
| N-Substituted Valiolamine Derivatives as Potent Inhibitors of Endoplasmic Reticulum α-Glucosidases I and II with Antiviral Activity. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |