| Assay ID | Title | Year | Journal | Article |
|---|
| AID219779 | Direct activation of chloride currents (percentage of 10 mM GABA response) in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunits | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID447576 | Binding affinity to apoferritin by isothermal titration calorimetry | 2009 | Bioorganic & medicinal chemistry, Jul-15, Volume: 17, Issue:14
| Structure-based shape pharmacophore modeling for the discovery of novel anesthetic compounds. |
| AID219780 | Modulation of GABA-induced chloride currents (percentage of GABA EC20 response) against human alpha-1-beta-1-gamma-2 GABA-A receptor subunits expressed in Xenopus laevis oocytes | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID71848 | Inhibition of [35S]TBPS binding to GABA-A receptor in rat cerebral cortex. | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID219778 | Modulation of GABA-induced chloride currents in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunits | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID15880 | Calculated partition coefficient (clogP) | 2002 | Journal of medicinal chemistry, Jul-18, Volume: 45, Issue:15
| 4D-QSAR analysis of a set of propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. |
| AID219644 | Direct activation of chloride current in Xenopus laevis oocytes expressing human alpha-1-beta-1-gamma-2 GABA-A receptor subunits | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID72642 | Potentiation of GABA responses at human Gamma-aminobutyric acid A receptor alpha-1-beta-2-gamma-2 | 2002 | Journal of medicinal chemistry, Jul-18, Volume: 45, Issue:15
| 4D-QSAR analysis of a set of propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. |
| AID19624 | Partition coefficient (logP) | 1998 | Journal of medicinal chemistry, May-21, Volume: 41, Issue:11
| Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. |
| AID72641 | Direct activation of human Gamma-aminobutyric acid A receptor alpha-1-beta-2-gamma-2 | 2002 | Journal of medicinal chemistry, Jul-18, Volume: 45, Issue:15
| 4D-QSAR analysis of a set of propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. |
| AID219760 | Loss of righting reflex (LORR) in Xenopus laevis tadpoles was determined for anesthetic activity | 2002 | Journal of medicinal chemistry, Jul-18, Volume: 45, Issue:15
| 4D-QSAR analysis of a set of propofol analogues: mapping binding sites for an anesthetic phenol on the GABA(A) receptor. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |