| Assay ID | Title | Year | Journal | Article |
|---|
| AID706377 | Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as blockade of Cl-IB-MECA-mediated inhibition of forskolin-stimulated [3H]cAMP accumulation by scintillation counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID34880 | Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cells | 2001 | Journal of medicinal chemistry, Mar-01, Volume: 44, Issue:5
| Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists. |
| AID706387 | Displacement of [3H]CCPA from rat adenosine A1 receptor expressed in CHO cells after 60 mins by gamma counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID34704 | Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cells | 2001 | Journal of medicinal chemistry, Nov-22, Volume: 44, Issue:24
| Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides. |
| AID706385 | Displacement of [125I]I-AB-MECA from human rat adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID143442 | Antimycoplasmal activity against Mycoplasma gallisepticum K514 with the extra addition of copper (40 uM) | 1988 | Journal of medicinal chemistry, Apr, Volume: 31, Issue:4
| Synthesis and copper-dependent antimycoplasmal activity of 1-amino-3-(2-pyridyl)isoquinoline derivatives. 1. Amides. |
| AID143566 | Antimycoplasmal activity against Mycoplasma gallisepticum K514 without the extra addition of copper | 1988 | Journal of medicinal chemistry, Apr, Volume: 31, Issue:4
| Synthesis and copper-dependent antimycoplasmal activity of 1-amino-3-(2-pyridyl)isoquinoline derivatives. 1. Amides. |
| AID706384 | Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID706389 | Displacement of [3H]CGS21680 from rat adenosine A2A receptor expressed in CHO cells after 60 mins by gamma counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID34867 | Tested for antagonist activity by displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| A novel class of adenosine A3 receptor ligands. 2. Structure affinity profile of a series of isoquinoline and quinazoline compounds. |
| AID706380 | Selectivity ratio of Ki for human recombinant adenosine A2A receptor to Ki for human recombinant adenosine A3 receptor expressed in CHO cells | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID34581 | Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cells | 2001 | Journal of medicinal chemistry, Nov-22, Volume: 44, Issue:24
| Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides. |
| AID33025 | Antagonistic activity assayed by displacement of specific [3H]-CGS-21,680 binding in rat striatal membrane (adenosine A2A receptor) at a conc of 10 mM. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| A novel class of adenosine A3 receptor ligands. 2. Structure affinity profile of a series of isoquinoline and quinazoline compounds. |
| AID32653 | Antagonist activity by displacement of specific [3H]DPCPX binding in rat cortical membrane (Adenosine A1 receptor) at a Conc of 10 mM. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| A novel class of adenosine A3 receptor ligands. 2. Structure affinity profile of a series of isoquinoline and quinazoline compounds. |
| AID32891 | Displacement of [3H]-CGS- 21680 binding in adenosine A2A receptor of rat striatal membrane | 2001 | Journal of medicinal chemistry, Mar-01, Volume: 44, Issue:5
| Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists. |
| AID32354 | Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membrane | 2001 | Journal of medicinal chemistry, Mar-01, Volume: 44, Issue:5
| Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists. |
| AID34995 | Percent displacement of [3H]-CGS- 21680 binding in adenosine A2A receptor of rat striatal membrane at a concentration of 10 uM | 2001 | Journal of medicinal chemistry, Mar-01, Volume: 44, Issue:5
| Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists. |
| AID706382 | Selectivity ratio of Ki for human recombinant adenosine A1 receptor to Ki for human recombinant adenosine A3 receptor expressed in CHO cells | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| AID268110 | Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cells | 2006 | Journal of medicinal chemistry, Jul-13, Volume: 49, Issue:14
| Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models. |
| AID32659 | Percent displacement of [3H]DPCPX binding in adenosine A1 receptor of rat brain cortical membrane at a concentration of 10 uM | 2001 | Journal of medicinal chemistry, Mar-01, Volume: 44, Issue:5
| Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists. |
| AID706386 | Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 60 mins by gamma counter | 2012 | Journal of medicinal chemistry, Jun-28, Volume: 55, Issue:12
| Medicinal chemistry of A₃ adenosine receptor modulators: pharmacological activities and therapeutic implications. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |