| Assay ID | Title | Year | Journal | Article |
|---|
| AID324626 | Intrinsic activity at human cloned 5HT2C receptor expressed in CHO cells assessed as maximal stimulation of 10 uM 5HT-induced myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324625 | Agonist activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326605 | Selectivity for human 5HT2C receptor over human 5HT2A receptor | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID326608 | Intrinsic activity at human 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol turnover relative to 5-hydroxytryptamine | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324622 | Selectivity for human 5HT2A to human 5HT2C | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324629 | Selectivity ratio of EC50 for human cloned 5HT2C receptor over EC50 for human cloned 5HT2A receptor | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324620 | Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cells | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326610 | Effect on 5-HT2A-mediated penile erection in rat | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324630 | Selectivity ratio of EC50 for human cloned 5HT2B receptor over EC50 for human cloned 5HT2C receptor | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326604 | Displacement of [3H]5-HT from human 5HT2B receptor expressed in HEK293-EBNA cells | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID326606 | Selectivity for human 5HT2C receptor over human 5HT2B receptor | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324621 | Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cells | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326607 | Intrinsic activity at human 5HT2C receptor expressed in CHO cells assessed as myo-[3H]inositol turnover relative to 5-hydroxytryptamine | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID326602 | Displacement of [3H]5-HT from human 5HT2C receptor expressed in CHO cells | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID326603 | Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cells | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324627 | Intrinsic activity at human cloned 5HT2A receptor expressed in CHO cells assessed as maximal stimulation of 10 uM 5HT-induced myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324631 | Induction of penile erection in sc dosed rat | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324632 | Induction of penile erection in po dosed rat | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID324628 | Intrinsic activity at human cloned 5HT2B receptor expressed in HEK293-EBNA cells assessed as maximal stimulation of 10 uM 5HT-induced myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326609 | Effect on 5-HT2C-mediated penile erection in rat | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324624 | Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326612 | Cardiovascular effect in po dosed rat assessed as increase in mean arterial blood pressure | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID324623 | Agonist activity at human cloned 5HT2C receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysis | 2008 | Bioorganic & medicinal chemistry, Feb-15, Volume: 16, Issue:4
| Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists. |
| AID326611 | Effect on penile erection in po dosed rat | 2008 | Bioorganic & medicinal chemistry, Mar-15, Volume: 16, Issue:6
| Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists. |
| AID624216 | Agonists at Human 5-Hydroxytryptamine receptor 5-HT2C | 2004 | European journal of pharmacology, Jan-01, Volume: 483, Issue:1
| Pharmacological profile of YM348, a novel, potent and orally active 5-HT2C receptor agonist. |
| AID1346893 | Human 5-HT2C receptor (5-Hydroxytryptamine receptors) | 2004 | European journal of pharmacology, Jan-01, Volume: 483, Issue:1
| Pharmacological profile of YM348, a novel, potent and orally active 5-HT2C receptor agonist. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |