| Assay ID | Title | Year | Journal | Article |
|---|
| AID1533312 | Potency index, ratio of tetrahydrolipstatin IC50 to compound IC50 for inhibition of ABHD16A (unknown origin) | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1533320 | Inhibition of TAMRA-FP binding to ABHD16A in rat cerebellar membranes at 10 uM preincubated for 1 hr followed by TAMRA-FP addition measured after 1 hr by fluorescence based ABPP analysis | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1533318 | Ratio of IC50 for reversible inhibition of human ABHD16A expressed in HEK293 cells to IC50 for inhibition of human ABHD16A expressed in HEK293 cells | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1533322 | Binding affinity to LYPLA1 in rat cerebellar membranes at 10 uM measured after 1 hr by fluorescence based ABPP analysis | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1533311 | Inhibition of ABHD16A (unknown origin) | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1533315 | Inhibition of human ABHD16A expressed in HEK293 cells preincubated for 30 mins followed by 1-LG substrate addition and measured after 90 to 120 mins by fluorometric assay | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID1079563 | Inhibition of APT1 (unknown origin) | 2014 | MedChemComm, Mar, Volume: 5, Issue:3
| Acyl protein thioesterase inhibitors as probes of dynamic S-palmitoylation. |
| AID1079562 | Inhibition of APT2 (unknown origin) | 2014 | MedChemComm, Mar, Volume: 5, Issue:3
| Acyl protein thioesterase inhibitors as probes of dynamic S-palmitoylation. |
| AID1533323 | Binding affinity to LYPLA2 in rat cerebellar membranes at 10 uM measured after 1 hr by fluorescence based ABPP analysis | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| AID576610 | Inhibition of APT1 | 2011 | Bioorganic & medicinal chemistry, Feb-15, Volume: 19, Issue:4
| Small molecule inhibition of protein depalmitoylation as a new approach towards downregulation of oncogenic Ras signalling. |
| AID1533316 | Reversible inhibition of human ABHD16A expressed in HEK293 cells preincubated for 30 mins followed by 40 fold compound dilution and subsequent 1-LG substrate addition and measured at 30 mins time interval for 120 mins by fluorometric assay | 2018 | ACS medicinal chemistry letters, Dec-13, Volume: 9, Issue:12
| Discovery of 12-Thiazole Abietanes as Selective Inhibitors of the Human Metabolic Serine Hydrolase hABHD16A. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |