| Assay ID | Title | Year | Journal | Article |
|---|
| AID1501058 | Inhibition of Porphyromonas gingivalis N-terminal His-tagged DPP4 expressed in Escherichia coli using Gly-Pro-p-nitroanilide as substrate | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID343975 | Inhibition of DPP2 | 2008 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 18, Issue:14
| Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads. |
| AID270815 | Inhibition of DPP2 | 2006 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 16, Issue:18
| Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines. |
| AID611366 | Inhibition of DPP2 | 2011 | Journal of medicinal chemistry, Aug-25, Volume: 54, Issue:16
| Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal? |
| AID56227 | Inhibition of human Dipeptidylpeptidase IV (DPP IV) | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors. |
| AID1501063 | Inhibition of bovine DPP9 | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID343973 | Inhibition of DPP9 | 2008 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 18, Issue:14
| Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads. |
| AID270817 | Selectivity for DPP2 over DPP4 | 2006 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 16, Issue:18
| Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines. |
| AID611365 | Inhibition of DPP4 | 2011 | Journal of medicinal chemistry, Aug-25, Volume: 54, Issue:16
| Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal? |
| AID611364 | Inhibition of DPP9 | 2011 | Journal of medicinal chemistry, Aug-25, Volume: 54, Issue:16
| Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal? |
| AID235301 | Ratio of IC50 for DPP IV to that of IC50 for DPP II | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors. |
| AID611363 | Inhibition of DPP8 | 2011 | Journal of medicinal chemistry, Aug-25, Volume: 54, Issue:16
| Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal? |
| AID1501062 | Inhibition of DPP8 (unknown origin) | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID1501061 | Inhibition of human DPP4 | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID56221 | Inhibition of human Dipeptidylpeptidase II (DPP II) | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors. |
| AID343972 | Inhibition of DPP8 | 2008 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 18, Issue:14
| Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads. |
| AID343974 | Inhibition of DPP4 | 2008 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 18, Issue:14
| Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 1: identification of dipeptide derived leads. |
| AID270818 | Selectivity for DPP2 over DPP8 | 2006 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 16, Issue:18
| Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines. |
| AID270816 | Inhibition of DPP8 | 2006 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 16, Issue:18
| Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines. |
| AID270814 | Inhibition of DPP4 | 2006 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 16, Issue:18
| Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines. |
| AID1501064 | Inhibition of DPP2 (unknown origin) | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID1501056 | Inhibition of Porphyromonas gingivalis N-terminal His-tagged DPP4 expressed in Escherichia coli at 10 uM using Gly-Pro-p-nitroanilide as substrate relative to control | 2017 | European journal of medicinal chemistry, Oct-20, Volume: 139 | Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1345410 | Human Dipeptidyl-peptidase 7 (S28: Lysosomal Pro-Xaa carboxypeptidase) | 2006 | Biochemical pharmacology, Jun-28, Volume: 72, Issue:1
| Dipeptidyl peptidase II and leukocyte cell death. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |