| Assay ID | Title | Year | Journal | Article |
|---|
| AID71266 | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-6-beta-3-gamma-2 | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID219954 | Binding affinity against alpha-3-beta-3-gamma-2 GABAA/BzR receptor subtype. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID72132 | Binding affinity against Diazepam insensitive (DI) Gamma-aminobutyric acid A receptor | 1995 | Journal of medicinal chemistry, May-12, Volume: 38, Issue:10
| Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors. |
| AID233962 | Ratio of binding affinity against DI Bz receptor to that of DS Bz receptor | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors. |
| AID73089 | Binding affinity to human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-2-beta-3-gamma-2 | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID40379 | Binding affinity for Diazepam-Insensitive fraction of GABA-A benzodiazepine receptors | 1993 | Journal of medicinal chemistry, Apr-16, Volume: 36, Issue:8
| Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors. |
| AID219795 | It is the ratio of Ki value for alpha-1-beta-3-gamma-2 to that of alpha-5-beta-3-gamma-2 | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID73530 | Binding affinity for Gamma-aminobutyric acid A receptor alpha-5-beta-3-gamma-2 | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID40381 | Binding affinity for Diazepam-Sensitive fraction of GABA-A benzodiazepine receptors | 1993 | Journal of medicinal chemistry, Apr-16, Volume: 36, Issue:8
| Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors. |
| AID71268 | Binding affinity against Gamma-aminobutyric acid A receptor alpha-6-beta-3-gamma-2 | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID73523 | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-5-beta-3-gamma-2 | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID219794 | Binding affinity against alpha-1-beta-3-gamma-2 GABAA/BzR receptor subtype. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID232720 | Selectivity ratio of alpha1 beta-3 gamma2 GABA A / BzR and alpha5 beta-3 gamma2 GABA A / BzR | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID40377 | Binding affinity for Diazepam sensitive (DS) isoform of the benzodiazepine (Bz) binding site on GABAA receptors | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors. |
| AID73244 | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-3-beta-3-gamma-2 | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID40376 | Binding affinity for Diazepam insensitive (DI) isoform of the benzodiazepine (Bz) binding site on GABAA receptors | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors. |
| AID226435 | GABA shift ratio at Diazepam sensitive fraction of GABA-A benzodiazepine receptor | 1993 | Journal of medicinal chemistry, Apr-16, Volume: 36, Issue:8
| Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors. |
| AID72927 | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-1-beta-3-gamma-2 | 2000 | Journal of medicinal chemistry, Jan-13, Volume: 43, Issue:1
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. |
| AID219940 | Binding affinity tested against alpha-2-beta-3-gamma-2 GABAA/BzR receptor subtype. | 1998 | Journal of medicinal chemistry, Oct-08, Volume: 41, Issue:21
| Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar |
| AID72133 | Binding affinity against Diazepam sensitive (DS) Gamma-aminobutyric acid A receptor in rat cerebellum. | 1995 | Journal of medicinal chemistry, May-12, Volume: 38, Issue:10
| Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors. |
| AID234197 | Selectivity for Diazepam insensitive compared to sensitive GABA-A benzodiazepine receptor fractions | 1993 | Journal of medicinal chemistry, Apr-16, Volume: 36, Issue:8
| Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |