Page last updated: 2024-09-05

zg 63 and pwz-029

zg 63 has been researched along with pwz-029 in 3 studies

Compound Research Comparison

Studies
(zg 63)
Trials
(zg 63)
Recent Studies (post-2010)
(zg 63)
Studies
(pwz-029)
Trials
(pwz-029)
Recent Studies (post-2010) (pwz-029)
6001407

Protein Interaction Comparison

ProteinTaxonomyzg 63 (IC50)pwz-029 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.514
GABA theta subunitRattus norvegicus (Norway rat)0.514
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.514

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Harris, B; Liu, R; Skolnick, P; Zhang, P; Zhang, W1
Bennett, DW; Cook, JM; Gan, T; He, X; Huang, Q; Liu, R; McKernan, R; Zhang, P1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1

Other Studies

3 other study(ies) available for zg 63 and pwz-029

ArticleYear
Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors.
    Journal of medicinal chemistry, 1995, May-12, Volume: 38, Issue:10

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Diazepam; Male; Molecular Probes; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship

1995
Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar
    Journal of medicinal chemistry, 1998, Oct-08, Volume: 41, Issue:21

    Topics: Animals; Benzodiazepines; Cell Line; Crystallography, X-Ray; Humans; Ligands; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Regression Analysis; Structure-Activity Relationship

1998
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000