Assay ID | Title | Year | Journal | Article |
AID1067411 | Selectivity for mGlu4 receptor (unknown origin) over mGlu8 receptor (unknown origin) | 2014 | ACS medicinal chemistry letters, Feb-13, Volume: 5, Issue:2
| Qualification of LSP1-2111 as a Brain Penetrant Group III Metabotropic Glutamate Receptor Orthosteric Agonist. |
AID1067413 | Selectivity for mGlu4 receptor (unknown origin) over mGlu6 receptor (unknown origin) | 2014 | ACS medicinal chemistry letters, Feb-13, Volume: 5, Issue:2
| Qualification of LSP1-2111 as a Brain Penetrant Group III Metabotropic Glutamate Receptor Orthosteric Agonist. |
AID1455165 | Selectivity ratio of EC50 for mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium accumulation to EC50 for mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric | 2018 | Journal of medicinal chemistry, 03-08, Volume: 61, Issue:5
| Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. |
AID1455162 | Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium accumulation by Fluo-4 AM dye based fluorescence assay | 2018 | Journal of medicinal chemistry, 03-08, Volume: 61, Issue:5
| Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. |
AID1067412 | Selectivity for mGlu4 receptor (unknown origin) over mGlu7 receptor (unknown origin) | 2014 | ACS medicinal chemistry letters, Feb-13, Volume: 5, Issue:2
| Qualification of LSP1-2111 as a Brain Penetrant Group III Metabotropic Glutamate Receptor Orthosteric Agonist. |
AID1455160 | Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium accumulation by Fluo-4 AM dye based fluorescence assay | 2018 | Journal of medicinal chemistry, 03-08, Volume: 61, Issue:5
| Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. |
AID1455161 | Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium accumulation by Fluo-4 AM dye based fluorescence assay | 2018 | Journal of medicinal chemistry, 03-08, Volume: 61, Issue:5
| Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites. |
AID1346285 | Human mGlu4 receptor (Metabotropic glutamate receptors) | 2012 | FASEB journal : official publication of the Federation of American Societies for Experimental Biology, Apr, Volume: 26, Issue:4
| A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential. |
AID1346263 | Human mGlu7 receptor (Metabotropic glutamate receptors) | 2012 | FASEB journal : official publication of the Federation of American Societies for Experimental Biology, Apr, Volume: 26, Issue:4
| A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential. |
AID1346272 | Human mGlu6 receptor (Metabotropic glutamate receptors) | 2012 | FASEB journal : official publication of the Federation of American Societies for Experimental Biology, Apr, Volume: 26, Issue:4
| A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |