| Assay ID | Title | Year | Journal | Article |
|---|
| AID419045 | Inhibition of 6-His tagged Staphylococcus aureus recombinant sortase delta N24 expressed in Escherichia coli BL21 (DE3) | 2009 | Bioorganic & medicinal chemistry, Apr-01, Volume: 17, Issue:7
| Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform. |
| AID1225229 | Inhibition of recombinant his-tagged human pyruvate kinase M1 expressed in Escherichia coli BL-21(DE3) using PEP as substrate at 10 uM after 5 mins by L-LDH coupled assay relative to control | 2015 | Journal of natural products, Mar-27, Volume: 78, Issue:3
| Synthetic analogues of the marine bisindole deoxytopsentin: potent selective inhibitors of MRSA pyruvate kinase. |
| AID254837 | Inhibitory activity against Sortase A from Staphylococcus aureus | 2005 | Bioorganic & medicinal chemistry letters, Nov-15, Volume: 15, Issue:22
| Bis(indole) alkaloids as sortase A inhibitors from the sponge Spongosorites sp. |
| AID401678 | Cytotoxicity against human A549 cells after 48 hrs by SRB assay | 2005 | Journal of natural products, May, Volume: 68, Issue:5
| Cytotoxic bisindole alkaloids from a marine sponge Spongosorites sp. |
| AID255501 | Minimum inhibitory concentration against Staphylococcus aureus Newman strain | 2005 | Bioorganic & medicinal chemistry letters, Nov-15, Volume: 15, Issue:22
| Bis(indole) alkaloids as sortase A inhibitors from the sponge Spongosorites sp. |
| AID401681 | Cytotoxicity against human XF498 cells after 48 hrs by SRB assay | 2005 | Journal of natural products, May, Volume: 68, Issue:5
| Cytotoxic bisindole alkaloids from a marine sponge Spongosorites sp. |
| AID1225230 | Inhibition of recombinant his-tagged human pyruvate kinase M2 expressed in Escherichia coli BL-21(DE3) using PEP as substrate at 10 uM after 5 mins by L-LDH coupled assay relative to control | 2015 | Journal of natural products, Mar-27, Volume: 78, Issue:3
| Synthetic analogues of the marine bisindole deoxytopsentin: potent selective inhibitors of MRSA pyruvate kinase. |
| AID401682 | Cytotoxicity against human HCT15 cells after 48 hrs by SRB assay | 2005 | Journal of natural products, May, Volume: 68, Issue:5
| Cytotoxic bisindole alkaloids from a marine sponge Spongosorites sp. |
| AID401680 | Cytotoxicity against human SK-MEL-2 cells after 48 hrs by SRB assay | 2005 | Journal of natural products, May, Volume: 68, Issue:5
| Cytotoxic bisindole alkaloids from a marine sponge Spongosorites sp. |
| AID1225232 | Inhibition of recombinant his-tagged human pyruvate kinase L expressed in Escherichia coli BL-21(DE3) using PEP as substrate at 10 uM after 5 mins by L-LDH coupled assay relative to control | 2015 | Journal of natural products, Mar-27, Volume: 78, Issue:3
| Synthetic analogues of the marine bisindole deoxytopsentin: potent selective inhibitors of MRSA pyruvate kinase. |
| AID1225231 | Inhibition of recombinant his-tagged human pyruvate kinase R expressed in Escherichia coli BL-21(DE3) using PEP as substrate at 10 uM after 5 mins by L-LDH coupled assay relative to control | 2015 | Journal of natural products, Mar-27, Volume: 78, Issue:3
| Synthetic analogues of the marine bisindole deoxytopsentin: potent selective inhibitors of MRSA pyruvate kinase. |
| AID1225224 | Inhibition of recombinant his-tagged methicillin-resistant Staphylococcus aureus pyruvate kinase expressed in Escherichia coli BL-21(DE3) using PEP as substrate after 5 mins by L-LDH coupled assay | 2015 | Journal of natural products, Mar-27, Volume: 78, Issue:3
| Synthetic analogues of the marine bisindole deoxytopsentin: potent selective inhibitors of MRSA pyruvate kinase. |
| AID401679 | Cytotoxicity against human SKOV3 cells after 48 hrs by SRB assay | 2005 | Journal of natural products, May, Volume: 68, Issue:5
| Cytotoxic bisindole alkaloids from a marine sponge Spongosorites sp. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |