| Assay ID | Title | Year | Journal | Article |
|---|
| AID1263070 | Irreversible inhibition of AChE (unknown origin) | 2015 | Bioorganic & medicinal chemistry, Dec-15, Volume: 23, Issue:24
| Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin. |
| AID710296 | Inhibition of human recombinant pancreatic lipase expressed in Pichia pastoris at 200 molar excess compound concentration pre-incubated for 2 hrs with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID710299 | Inhibition of Fusarium solani pisi cutinase assessed as half inactivation time pre-incubated with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID1263069 | Inhibition of AChE (unknown origin) | 2015 | Bioorganic & medicinal chemistry, Dec-15, Volume: 23, Issue:24
| Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin. |
| AID1263068 | Inhibition of housefly CSMA AChE | 2015 | Bioorganic & medicinal chemistry, Dec-15, Volume: 23, Issue:24
| Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin. |
| AID710304 | Inhibition of Mycobacterium tuberculosis LipY pre-incubated for 30 mins with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID710303 | Inhibition of Mycobacterium tuberculosis LipY at 40 molar excess compound concentration pre-incubated for 30 mins with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID1263072 | Inhibition of human AChE at pH 6 | 2015 | Bioorganic & medicinal chemistry, Dec-15, Volume: 23, Issue:24
| Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin. |
| AID710294 | Inhibition of dog recombinant gastric lipase expressed in transgenic maize at 200 molar excess compound concentration pre-incubated for 2 hrs with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID710295 | Inhibition of guinea pig recombinant PLRP2 expressed in Aspergillus oryzae at 200 molar excess compound concentration pre-incubated for 2 hrs with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID710302 | Inhibition of Fusarium solani pisi cutinase assessed as residual enzyme activity pre-incubated for 30 mins with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID462370 | Inhibition of AChE by modified Ellman's spectrophotometric method | 2010 | Bioorganic & medicinal chemistry, Mar-15, Volume: 18, Issue:6
| Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase. |
| AID1263071 | Inhibition of human AChE at pH 8 | 2015 | Bioorganic & medicinal chemistry, Dec-15, Volume: 23, Issue:24
| Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin. |
| AID710305 | Inhibition of Mycobacterium tuberculosis Rv0183 pre-incubated for 30 mins with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| AID1192914 | Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation counting | 2015 | Bioorganic & medicinal chemistry, Mar-01, Volume: 23, Issue:5
| Rat hormone sensitive lipase inhibition by cyclipostins and their analogs. |
| AID710306 | Inhibition of Fusarium solani pisi cutinase pre-incubated for 30 mins with enzyme before substrate addition by pH-stat technique | 2012 | Journal of medicinal chemistry, Nov-26, Volume: 55, Issue:22
| Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |