| Assay ID | Title | Year | Journal | Article |
|---|
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1460830 | Inhibition of ABHD6 in mouse BV2 cells preincubated for 30 mins and subsequent addition of [3H]-2-OG substrate measured after 15 mins by liquid scintillation counting method | 2017 | Bioorganic & medicinal chemistry, 11-15, Volume: 25, Issue:22
| Biological evaluation of pyridone alkaloids on the endocannabinoid system. |
| AID1624798 | Inhibition of ABHD6 in mouse brain membrane assessed as protein band intensity at 10 uM pre-incubated for 25 mins followed by TAMRA-FP probe labeling for 5 mins by SDS-PAGE analysis relative to control | 2019 | Journal of medicinal chemistry, 02-28, Volume: 62, Issue:4
| Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible Monoacylglycerol Lipase (MAGL) Inhibitor. |
| AID1460831 | Inhibition of ABHD12 in mouse BV2 cells preincubated for 30 mins and subsequent addition of [3H]-2-OG substrate measured after 15 mins by liquid scintillation counting method | 2017 | Bioorganic & medicinal chemistry, 11-15, Volume: 25, Issue:22
| Biological evaluation of pyridone alkaloids on the endocannabinoid system. |
| AID1910304 | Inhibition of ABHD6 in mouse brain membrane at 10 uM using TAMRA-FP serine hydrolase probe as substrate preincubated for 25 mins followed by substrate addition and measured after 25 mins SDS-PAGE analysis | 2022 | Journal of medicinal chemistry, 05-26, Volume: 65, Issue:10
| Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives. |
| AID1624796 | Inhibition of FAAH in mouse brain membrane assessed as protein band intensity at 10 uM pre-incubated for 25 mins followed by TAMRA-FP probe labeling for 5 mins by SDS-PAGE analysis relative to control | 2019 | Journal of medicinal chemistry, 02-28, Volume: 62, Issue:4
| Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible Monoacylglycerol Lipase (MAGL) Inhibitor. |
| AID1624797 | Inhibition of MAGL in mouse brain membrane assessed as protein band intensity at 10 uM pre-incubated for 25 mins followed by TAMRA-FP probe labeling for 5 mins by SDS-PAGE analysis relative to control | 2019 | Journal of medicinal chemistry, 02-28, Volume: 62, Issue:4
| Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible Monoacylglycerol Lipase (MAGL) Inhibitor. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |