Page last updated: 2024-09-04

pumosetrag and cisapride

pumosetrag has been researched along with cisapride in 1 studies

Compound Research Comparison

Studies
(pumosetrag)
Trials
(pumosetrag)
Recent Studies (post-2010)
(pumosetrag)
Studies
(cisapride)
Trials
(cisapride)
Recent Studies (post-2010) (cisapride)
8431,554390110

Protein Interaction Comparison

ProteinTaxonomypumosetrag (IC50)cisapride (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.767
3-hydroxy-3-methylglutaryl-coenzyme A reductaseHomo sapiens (human)3.37
Cytochrome P450 3A4Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0098
Alpha-2A adrenergic receptorHomo sapiens (human)3.5923
Cytochrome P450 2D6Homo sapiens (human)0.07
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)0.1701
D(2) dopamine receptorHomo sapiens (human)0.35
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)2.69
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0098
Insulin receptor Rattus norvegicus (Norway rat)3.37
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)2.29
Alpha-2B adrenergic receptorHomo sapiens (human)3.3827
Alpha-2C adrenergic receptorHomo sapiens (human)3.26
DRattus norvegicus (Norway rat)0.0065
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.6495
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0065
D(1A) dopamine receptorHomo sapiens (human)1.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0065
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0065
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)2.29
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0065
Alpha-1D adrenergic receptorHomo sapiens (human)0.083
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0054
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.2597
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.6495
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)4.47
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)4.47
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0098
Sodium-dependent serotonin transporterHomo sapiens (human)0.384
Alpha-1A adrenergic receptorHomo sapiens (human)0.03
Prostaglandin G/H synthase 2Homo sapiens (human)3.37
Alpha-1B adrenergic receptorHomo sapiens (human)0.03
D(3) dopamine receptorHomo sapiens (human)0.144
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.9
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0407
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)2.29
D(2) dopamine receptorRattus norvegicus (Norway rat)0.535
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.2536
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)0.1701
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.994
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.9

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chai, W; Chan, KY; Danser, AH; de Maeyer, JH; de Vries, R; MaassenVanDenBrink, A; Saxena, PR; Schuurkes, JA; van den Bogeardt, AJ; Villalón, CM1

Other Studies

1 other study(ies) available for pumosetrag and cisapride

ArticleYear
Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.
    Life sciences, 2012, Apr-09, Volume: 90, Issue:13-14

    Topics: 5-Methoxytryptamine; Adolescent; Adult; Aged; Benzofurans; Calcium Channels; Child; Cisapride; Female; Gastrointestinal Agents; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Middle Aged; Muscle Contraction; Myocardium; Pyridines; Quinuclidines; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Sulfonamides; Young Adult

2012