Assay ID | Title | Year | Journal | Article |
AID215747 | Binding affinity against trypsin | 2004 | Bioorganic & medicinal chemistry letters, Jun-21, Volume: 14, Issue:12
| Interaction with the S1 beta-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors. |
AID419413 | Inhibition of urokinase | 2009 | Journal of medicinal chemistry, May-28, Volume: 52, Issue:10
| Large-scale application of high-throughput molecular mechanics with Poisson-Boltzmann surface area for routine physics-based scoring of protein-ligand complexes. |
AID158340 | Binding affinity against plasmin | 2004 | Bioorganic & medicinal chemistry letters, Jun-21, Volume: 14, Issue:12
| Interaction with the S1 beta-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors. |
AID150768 | Binding affinity towards P-kallikrein | 2004 | Bioorganic & medicinal chemistry letters, Jun-21, Volume: 14, Issue:12
| Interaction with the S1 beta-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors. |
AID210752 | Binding affinity towards human Tissue type plasminogen activator. | 2004 | Journal of medicinal chemistry, Jan-15, Volume: 47, Issue:2
| Identification of novel binding interactions in the development of potent, selective 2-naphthamidine inhibitors of urokinase. Synthesis, structural analysis, and SAR of N-phenyl amide 6-substitution. |
AID213441 | Binding affinity towards Urokinase-type plasminogen activator (urokinase) | 2004 | Bioorganic & medicinal chemistry letters, Jun-21, Volume: 14, Issue:12
| Interaction with the S1 beta-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors. |
AID210919 | Binding affinity towards tissue type plasminogen activator | 2004 | Bioorganic & medicinal chemistry letters, Jun-21, Volume: 14, Issue:12
| Interaction with the S1 beta-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors. |
AID157977 | Binding affinity towards human plasmin. | 2004 | Journal of medicinal chemistry, Jan-15, Volume: 47, Issue:2
| Identification of novel binding interactions in the development of potent, selective 2-naphthamidine inhibitors of urokinase. Synthesis, structural analysis, and SAR of N-phenyl amide 6-substitution. |
AID215587 | Binding affinity against porcine trypsin was determined. | 2004 | Journal of medicinal chemistry, Jan-15, Volume: 47, Issue:2
| Identification of novel binding interactions in the development of potent, selective 2-naphthamidine inhibitors of urokinase. Synthesis, structural analysis, and SAR of N-phenyl amide 6-substitution. |
AID215835 | Binding affinity to human urokinase-type plasminogen activator (microPa). | 2004 | Journal of medicinal chemistry, Jan-15, Volume: 47, Issue:2
| Identification of novel binding interactions in the development of potent, selective 2-naphthamidine inhibitors of urokinase. Synthesis, structural analysis, and SAR of N-phenyl amide 6-substitution. |
AID95041 | Binding affinity against human plasma kallikrein. | 2004 | Journal of medicinal chemistry, Jan-15, Volume: 47, Issue:2
| Identification of novel binding interactions in the development of potent, selective 2-naphthamidine inhibitors of urokinase. Synthesis, structural analysis, and SAR of N-phenyl amide 6-substitution. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |