| Assay ID | Title | Year | Journal | Article |
|---|
| AID656660 | Ratio of drug uptake in Alzheimer's disease patient brain to healthy human brain | 2011 | ACS medicinal chemistry letters, Sep-08, Volume: 2, Issue:9
| A Novel (18)F-Labeled Imidazo[2,1-b]benzothiazole (IBT) for High-Contrast PET Imaging of β-Amyloid Plaques. |
| AID695043 | Binding affinity to amyloid beta (1-42) aggregates | 2012 | Journal of medicinal chemistry, Jan-26, Volume: 55, Issue:2
| Synthesis and evaluation of ¹⁸F-labeled styryltriazole and resveratrol derivatives for β-amyloid plaque imaging. |
| AID438578 | Drug uptake in mouse brain after 60 mins | 2009 | Journal of medicinal chemistry, Oct-22, Volume: 52, Issue:20
| Fluoro-pegylated chalcones as positron emission tomography probes for in vivo imaging of beta-amyloid plaques in Alzheimer's disease. |
| AID623031 | Drug uptake in mouse brain | 2011 | Bioorganic & medicinal chemistry letters, Oct-01, Volume: 21, Issue:19
| Synthesis and evaluation of 1-(4-[¹⁸F]fluoroethyl)-7-(4'-methyl)curcumin with improved brain permeability for β-amyloid plaque imaging. |
| AID695088 | Partition coefficient, log P of the compound | 2012 | Journal of medicinal chemistry, Jan-26, Volume: 55, Issue:2
| Synthesis and evaluation of ¹⁸F-labeled styryltriazole and resveratrol derivatives for β-amyloid plaque imaging. |
| AID695087 | Ratio of drug uptake in mouse brain after 2 mins to 30 mins | 2012 | Journal of medicinal chemistry, Jan-26, Volume: 55, Issue:2
| Synthesis and evaluation of ¹⁸F-labeled styryltriazole and resveratrol derivatives for β-amyloid plaque imaging. |
| AID438579 | Drug uptake in mouse bone after 60 mins | 2009 | Journal of medicinal chemistry, Oct-22, Volume: 52, Issue:20
| Fluoro-pegylated chalcones as positron emission tomography probes for in vivo imaging of beta-amyloid plaques in Alzheimer's disease. |
| AID596273 | Ratio of drug level in brain after 2 mins to brain after 60 mins in ddY mouse heart at 185 to 370 kBq, iv | 2011 | Journal of medicinal chemistry, Apr-28, Volume: 54, Issue:8
| Novel 18F-labeled benzofuran derivatives with improved properties for positron emission tomography (PET) imaging of β-amyloid plaques in Alzheimer's brains. |
| AID706000 | Displacement of [125I]-IMPY from amyloid beta (1 to 42) fibrils after 2 hrs by gamma-counting analysis | 2012 | Journal of medicinal chemistry, Nov-08, Volume: 55, Issue:21
| Synthesis and evaluation of novel ¹⁸F labeled 2-pyridinylbenzoxazole and 2-pyridinylbenzothiazole derivatives as ligands for positron emission tomography (PET) imaging of β-amyloid plaques. |
| AID705778 | Drug uptake in iv dosed ICR mouse brain at 60 mins | 2012 | Journal of medicinal chemistry, Nov-08, Volume: 55, Issue:21
| Synthesis and evaluation of novel ¹⁸F labeled 2-pyridinylbenzoxazole and 2-pyridinylbenzothiazole derivatives as ligands for positron emission tomography (PET) imaging of β-amyloid plaques. |
| AID695045 | Drug uptake in mouse brain after 2 mins | 2012 | Journal of medicinal chemistry, Jan-26, Volume: 55, Issue:2
| Synthesis and evaluation of ¹⁸F-labeled styryltriazole and resveratrol derivatives for β-amyloid plaque imaging. |
| AID705788 | Drug uptake in iv dosed ICR mouse brain at 2 mins | 2012 | Journal of medicinal chemistry, Nov-08, Volume: 55, Issue:21
| Synthesis and evaluation of novel ¹⁸F labeled 2-pyridinylbenzoxazole and 2-pyridinylbenzothiazole derivatives as ligands for positron emission tomography (PET) imaging of β-amyloid plaques. |
| AID705789 | Ratio of drug uptake in brain at 2 mins to drug uptake in brain at 60 mins in iv dosed ICR mouse | 2012 | Journal of medicinal chemistry, Nov-08, Volume: 55, Issue:21
| Synthesis and evaluation of novel ¹⁸F labeled 2-pyridinylbenzoxazole and 2-pyridinylbenzothiazole derivatives as ligands for positron emission tomography (PET) imaging of β-amyloid plaques. |
| AID755102 | Displacement of [125I]IMPY from amyloid beta in brain homogenate of Alzheimer's disease patient after 2 hrs by gamma counting analysis | 2013 | Bioorganic & medicinal chemistry, Jul-01, Volume: 21, Issue:13
| Synthesis and biological evaluation of 18F-labled 2-phenylindole derivatives as PET imaging probes for β-amyloid plaques. |
| AID673978 | Binding affinity to human amyloid beta plaque | 2012 | ACS medicinal chemistry letters, Apr-12, Volume: 3, Issue:4
| The β-Amyloid Hypothesis in Alzheimer's Disease: Seeing Is Believing. |
| AID438577 | Drug uptake in mouse brain after 2 mins | 2009 | Journal of medicinal chemistry, Oct-22, Volume: 52, Issue:20
| Fluoro-pegylated chalcones as positron emission tomography probes for in vivo imaging of beta-amyloid plaques in Alzheimer's disease. |
| AID695046 | Binding affinity to amyloid beta (1-42) aggregates in human Alzheimer's disease brain sections | 2012 | Journal of medicinal chemistry, Jan-26, Volume: 55, Issue:2
| Synthesis and evaluation of ¹⁸F-labeled styryltriazole and resveratrol derivatives for β-amyloid plaque imaging. |
| AID684724 | Binding affinity to beta-amyloid | 2012 | European journal of medicinal chemistry, Nov, Volume: 57 | ¹⁸F-labeled 2-phenylquinoxaline derivatives as potential positron emission tomography probes for in vivo imaging of β-amyloid plaques. |
| AID438576 | Binding affinity to amyloid beta (1 to 42) peptide | 2009 | Journal of medicinal chemistry, Oct-22, Volume: 52, Issue:20
| Fluoro-pegylated chalcones as positron emission tomography probes for in vivo imaging of beta-amyloid plaques in Alzheimer's disease. |
| AID668927 | Displacement of [18F]-amyvid from amyloid-beta aggregates in alzheimer's disease patient brain homogenates after 1 hr | 2011 | Journal of medicinal chemistry, Dec-08, Volume: 54, Issue:23
| Multidentate (18)F-polypegylated styrylpyridines as imaging agents for Aβ plaques in cerebral amyloid angiopathy (CAA). |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |