Page last updated: 2024-09-05

bd 1047 and donepezil

bd 1047 has been researched along with donepezil in 2 studies

Compound Research Comparison

Studies
(bd 1047)
Trials
(bd 1047)
Recent Studies (post-2010)
(bd 1047)
Studies
(donepezil)
Trials
(donepezil)
Recent Studies (post-2010) (donepezil)
1180543,1935571,594

Protein Interaction Comparison

ProteinTaxonomybd 1047 (IC50)donepezil (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.4231
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.0265
Amyloid-beta precursor proteinHomo sapiens (human)0.022
CholinesteraseHomo sapiens (human)4.5742
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.42
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)5
Amine oxidase [flavin-containing] A Rattus norvegicus (Norway rat)7.4
AcetylcholinesteraseMus musculus (house mouse)1.5489
AcetylcholinesteraseHomo sapiens (human)0.3257
Acetylcholinesterase Bos taurus (cattle)0.1644
Choline O-acetyltransferase Rattus norvegicus (Norway rat)0.0053
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0182
Beta-secretase 1Homo sapiens (human)0.8666
CholinesteraseEquus caballus (horse)3.7325
CholinesteraseMus musculus (house mouse)1.992
Acetylcholine receptor subunit epsilonHomo sapiens (human)0.0324
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.7844
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.008
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)4.715
Carboxylic ester hydrolase Equus caballus (horse)4.5551
Histamine H3 receptorHomo sapiens (human)0.35

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Feng, B; Ieni, J; Maurice, T; Meunier, J; Monaghan, DT1
Ieni, J; Maurice, T; Meunier, J1

Other Studies

2 other study(ies) available for bd 1047 and donepezil

ArticleYear
Interaction with sigma(1) protein, but not N-methyl-D-aspartate receptor, is involved in the pharmacological activity of donepezil.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 317, Issue:2

    Topics: Animals; Avoidance Learning; Behavior, Animal; Binding Sites; Cholinesterase Inhibitors; Cloning, Molecular; Donepezil; Ethylenediamines; Female; Indans; Ligands; Male; Maze Learning; Mice; Oligodeoxyribonucleotides, Antisense; Oocytes; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Swimming; Xenopus

2006
The anti-amnesic and neuroprotective effects of donepezil against amyloid beta25-35 peptide-induced toxicity in mice involve an interaction with the sigma1 receptor.
    British journal of pharmacology, 2006, Volume: 149, Issue:8

    Topics: Amnesia; Amyloid beta-Peptides; Animals; Avoidance Learning; Behavior, Animal; Donepezil; Dose-Response Relationship, Drug; Ethylenediamines; Fluorescent Dyes; Galantamine; Indans; Injections, Intraventricular; Lipid Peroxidation; Male; Maze Learning; Mice; Neuroprotective Agents; Nootropic Agents; Peptide Fragments; Phenols; Phenylcarbamates; Piperidines; Receptors, sigma; Rivastigmine; Sulfoxides; Xylenes

2006