Page last updated: 2024-09-05

ahr-2666 and verapamil

ahr-2666 has been researched along with verapamil in 3 studies

Compound Research Comparison

Studies
(ahr-2666)
Trials
(ahr-2666)
Recent Studies (post-2010)
(ahr-2666)
Studies
(verapamil)
Trials
(verapamil)
Recent Studies (post-2010) (verapamil)
50017,6211,5272,067

Protein Interaction Comparison

ProteinTaxonomyahr-2666 (IC50)verapamil (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)6.8
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.2
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
ATP-dependent translocase ABCB1Mus musculus (house mouse)2
ATP-dependent translocase ABCB1Homo sapiens (human)2.2346
Cytochrome P450 3A4Homo sapiens (human)3.8008
Alpha-2A adrenergic receptorHomo sapiens (human)0.579
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.02
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
Catechol O-methyltransferaseHomo sapiens (human)0.2
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)8
Histamine H2 receptorHomo sapiens (human)2.59
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.442
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.02
Sodium-dependent serotonin transporterHomo sapiens (human)0.24
Multidrug resistance-associated protein 1 Homo sapiens (human)5.598
D(3) dopamine receptorHomo sapiens (human)0.186
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.165
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)6.8
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.2
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.3945
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.2
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.175
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.1934

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19903 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Danilo, P; Davies, M; Hordof, AJ; Reder, RF; Rosen, MR1
Danilo, P; Rosen, MR1
Danilo, P; Hordof, AJ; Malm, JR; Mary-Rabine, L; Rosen, MR1

Other Studies

3 other study(ies) available for ahr-2666 and verapamil

ArticleYear
Age-related changes in Purkinje fiber action potentials of adult dogs.
    Circulation research, 1978, Volume: 43, Issue:6

    Topics: Action Potentials; Aging; Animals; Carbamates; Dogs; Electrocardiography; Female; Heart Conduction System; Male; Microelectrodes; Purkinje Fibers; Pyrrolidines; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1978
Effects of tetrodotoxin, lidocaine, verapamil, and AHR-2666 on Ouabain-induced delayed afterdepolarizations in canine Purkinje fibers.
    Circulation research, 1980, Volume: 46, Issue:1

    Topics: Action Potentials; Animals; Carbamates; Diastole; Dogs; Heart Conduction System; Ion Channels; Lidocaine; Ouabain; Purkinje Fibers; Pyrrolidines; Tetrodotoxin; Time Factors; Verapamil

1980
Mechanisms for impulse initiation in isolated human atrial fibers.
    Circulation research, 1980, Volume: 47, Issue:2

    Topics: Acetylcholine; Action Potentials; Adolescent; Adult; Carbamates; Child; Child, Preschool; Electrophysiology; Epinephrine; Heart Atria; Heart Conduction System; Heart Rate; Humans; Infant; Lidocaine; Middle Aged; Myocardial Contraction; Pyrrolidines; Tetrodotoxin; Time Factors; Verapamil

1980