| Assay ID | Title | Year | Journal | Article |
|---|
| AID141119 | Inhibitory activity against muscle Glycogen Phosphorylase b | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Synthesis of and a comparative study on the inhibition of muscle and liver glycogen phosphorylases by epimeric pairs of d-gluco- and d-xylopyranosylidene-spiro-(thio)hydantoins and N-(d-glucopyranosyl) amides. |
| AID1276749 | Competitive inhibition of rabbit skeletal muscle glycogen phosphorylase b | 2016 | European journal of medicinal chemistry, Jan-27, Volume: 108 | Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition. |
| AID141117 | Inhibitory activity against liver Glycogen Phosphorylase b | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Synthesis of and a comparative study on the inhibition of muscle and liver glycogen phosphorylases by epimeric pairs of d-gluco- and d-xylopyranosylidene-spiro-(thio)hydantoins and N-(d-glucopyranosyl) amides. |
| AID141233 | Inhibitor constant was measured against Muscle phosphorylase b in rabbit | 1999 | Bioorganic & medicinal chemistry letters, May-17, Volume: 9, Issue:10
| Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin. |
| AID141231 | Inhibitor constant was measured against Muscle phosphorylase a in rabbit | 1999 | Bioorganic & medicinal chemistry letters, May-17, Volume: 9, Issue:10
| Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin. |
| AID101995 | Inhibitor constant was measured against Liver phosphorylase a in rat | 1999 | Bioorganic & medicinal chemistry letters, May-17, Volume: 9, Issue:10
| Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin. |
| AID644850 | Inhibition of rabbit muscle glycogen phosphorylase b assessed as inorganic phosphate release at pH 6.8 | 2012 | Bioorganic & medicinal chemistry, Mar-01, Volume: 20, Issue:5
| N-(4-Substituted-benzoyl)-N'-(β-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods. |
| AID101852 | Inhibitory activity against muscle Glycogen Phosphorylase a | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Synthesis of and a comparative study on the inhibition of muscle and liver glycogen phosphorylases by epimeric pairs of d-gluco- and d-xylopyranosylidene-spiro-(thio)hydantoins and N-(d-glucopyranosyl) amides. |
| AID453252 | Inhibition of rabbit muscle glycogen phosphorylase b | 2009 | Bioorganic & medicinal chemistry, Oct-15, Volume: 17, Issue:20
| Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors. |
| AID101996 | Inhibitor constant was measured against Liver phosphorylase b in rat | 1999 | Bioorganic & medicinal chemistry letters, May-17, Volume: 9, Issue:10
| Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin. |
| AID101851 | Inhibitory activity against liver Glycogen Phosphorylase a | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Synthesis of and a comparative study on the inhibition of muscle and liver glycogen phosphorylases by epimeric pairs of d-gluco- and d-xylopyranosylidene-spiro-(thio)hydantoins and N-(d-glucopyranosyl) amides. |
| AID387864 | Inhibition of rabbit muscle glycogen phosphorylase b | 2008 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 18, Issue:20
| Novel design principle validated: glucopyranosylidene-spiro-oxathiazole as new nanomolar inhibitor of glycogen phosphorylase, potential antidiabetic agent. |
| AID1563539 | Inhibition of rabbit muscle Glycogen phosphorylase b using glucose-1-phosphate as substrate in presence of AMP | 2019 | Journal of medicinal chemistry, 07-11, Volume: 62, Issue:13
| Glucopyranosylidene-spiro-imidazolinones, a New Ring System: Synthesis and Evaluation as Glycogen Phosphorylase Inhibitors by Enzyme Kinetics and X-ray Crystallography. |
| AID1280560 | Inhibition of rat liver glycogen phosphorylase | 2015 | ACS medicinal chemistry letters, Dec-10, Volume: 6, Issue:12
| 4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase. |
| AID977610 | Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB | 2002 | Bioorganic & medicinal chemistry, Feb, Volume: 10, Issue:2
| Kinetic and crystallographic studies of glucopyranosylidene spirothiohydantoin binding to glycogen phosphorylase B. |
| AID1811 | Experimentally measured binding affinity data derived from PDB | 2002 | Bioorganic & medicinal chemistry, Feb, Volume: 10, Issue:2
| Kinetic and crystallographic studies of glucopyranosylidene spirothiohydantoin binding to glycogen phosphorylase B. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |