Assay ID | Title | Year | Journal | Article |
AID1333330 | Competitive inhibition of rabbit muscle glycogen phosphorylase-b in presence of varying levels of glucose-1-phosphate and constant concentration of glycogen and AMP by double reciprocal plot method | 2016 | European journal of medicinal chemistry, Nov-10, Volume: 123 | Synthetic, enzyme kinetic, and protein crystallographic studies of C-β-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase. |
AID1280561 | Competitive inhibition of rabbit muscle glycogen phosphorylase-b using glucose-1-phosphate as substrate preincubated with glycogen for 15 mins followed by substrate addition measured every 1 min for 5 mins | 2015 | ACS medicinal chemistry letters, Dec-10, Volume: 6, Issue:12
| 4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase. |
AID1321911 | Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by double-reciprocal plot analysis | 2016 | Bioorganic & medicinal chemistry, 11-01, Volume: 24, Issue:21
| Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitors. |
AID760348 | Inhibition of rabbit muscle glycogen phosphorylase b | 2013 | ACS medicinal chemistry letters, Jul-11, Volume: 4, Issue:7
| C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase. |
AID1333332 | Inhibition of rabbit muscle glycogen phosphorylase-b | 2016 | European journal of medicinal chemistry, Nov-10, Volume: 123 | Synthetic, enzyme kinetic, and protein crystallographic studies of C-β-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase. |
AID1280562 | Inhibition of rabbit muscle glycogen phosphorylase-b | 2015 | ACS medicinal chemistry letters, Dec-10, Volume: 6, Issue:12
| 4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase. |
AID1452109 | Competitive inhibition of rabbit muscle glycogen phosphorylase b using glucose-1-phosphate as substrate in presence of constant concentrations of glycogen and AMP | 2017 | Journal of medicinal chemistry, 11-22, Volume: 60, Issue:22
| Nanomolar Inhibitors of Glycogen Phosphorylase Based on β-d-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study. |
AID427132 | Inhibition of rabbit muscle glycogen phosphorylase b | 2009 | Bioorganic & medicinal chemistry, Jul-01, Volume: 17, Issue:13
| Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase. |
AID661299 | Binding affinity to rabbit muscular GPb by NMR binding assay | 2012 | Journal of medicinal chemistry, Feb-09, Volume: 55, Issue:3
| Binding evaluation of fragment-based scaffolds for probing allosteric enzymes. |
AID1129610 | Inhibition of rabbit muscle glycogen phosphorylase b | 2014 | European journal of medicinal chemistry, Apr-09, Volume: 76 | New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase. |
AID1321910 | Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrate | 2016 | Bioorganic & medicinal chemistry, 11-01, Volume: 24, Issue:21
| Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |