| Assay ID | Title | Year | Journal | Article |
|---|
| AID276213 | Effect on carrageenan-induced paw hyperalgesia in po dosed rat | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276218 | Binding affinity to TP receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276202 | Binding affinity to EP3 receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276217 | Binding affinity to IP receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276216 | Cmax in Sprague-Dawley rat at 10 mg/kg, po and 5 mg/kg, iv after 1 hr | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276204 | Antagonistic activity at EP3 receptor assessed as inhibition of cAMP production in HEK EBNA cells | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276208 | Bioavailability in Sprague-Dawley rat at 10 mg/kg, po and 5 mg/kg, iv | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276209 | Clearance in Sprague-Dawley rat at 10 mg/kg, po and 5 mg/kg, iv | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276220 | Binding affinity to DP receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276214 | Concentration in carrageenan-induced hyperalgesic rat at 10 mg/kg, po, 1 hr postdose | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276212 | Antiinflammatory activity against carrageenan-induced paw edema in po dosed rat | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276219 | Binding affinity to FP receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276201 | Binding affinity to EP2 receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276205 | Stability in rat hepatocytes after 3 hrs | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276200 | Binding affinity to EP1 receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276221 | Binding affinity to EP3 receptor in presence of HSA | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276207 | Metabolism in human hepatocytes | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276210 | Half life in Sprague-Dawley rat at 10 mg/kg, po and 5 mg/kg, iv | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID276203 | Binding affinity to EP4 receptor | 2006 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 16, Issue:21
| Comparison between two classes of selective EP(3) antagonists and their biological activities. |
| AID1347153 | Confirmatory screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347057 | CD47-SIRPalpha protein protein interaction - LANCE assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
| AID1347152 | Confirmatory screen NINDS AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347167 | Vero cells viability qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347151 | Optimization of GU AMC qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347410 | qHTS for inhibitors of adenylyl cyclases using a fission yeast platform: a pilot screen against the NCATS LOPAC library | 2019 | Cellular signalling, 08, Volume: 60 | A fission yeast platform for heterologous expression of mammalian adenylyl cyclases and high throughput screening. |
| AID1347058 | CD47-SIRPalpha protein protein interaction - HTRF assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
| AID1347405 | qHTS to identify inhibitors of the type 1 interferon - major histocompatibility complex class I in skeletal muscle: primary screen against the NCATS LOPAC collection | 2020 | ACS chemical biology, 07-17, Volume: 15, Issue:7
| High-Throughput Screening to Identify Inhibitors of the Type I Interferon-Major Histocompatibility Complex Class I Pathway in Skeletal Muscle. |
| AID1347149 | Furin counterscreen qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347169 | Tertiary RLuc qRT-PCR qHTS assay for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347161 | Confirmatory screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347059 | CD47-SIRPalpha protein protein interaction - Alpha assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
| AID1347168 | HepG2 cells viability qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347164 | 384 well plate NINDS Rhodamine confirmatory qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347163 | 384 well plate NINDS AMC confirmatory qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347156 | DAPI mCherry counterscreen qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347158 | ZIKV-mCherry secondary qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1346343 | Human EP3 receptor (Prostanoid receptors) | 2009 | British journal of pharmacology, Sep, Volume: 158, Issue:1
| Dual modulation of urinary bladder activity and urine flow by prostanoid EP3 receptors in the conscious rat. |
| AID1346343 | Human EP3 receptor (Prostanoid receptors) | 2001 | Bioorganic & medicinal chemistry, Aug, Volume: 9, Issue:8
| Structure-activity relationship of cinnamic acylsulfonamide analogues on the human EP3 prostanoid receptor. |
| AID1346343 | Human EP3 receptor (Prostanoid receptors) | 2008 | American journal of physiology. Renal physiology, Oct, Volume: 295, Issue:4
| Modulation of bladder function by prostaglandin EP3 receptors in the central nervous system. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | 2014 | Journal of biomolecular screening, Jul, Volume: 19, Issue:6
| A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | | | |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |