| Assay ID | Title | Year | Journal | Article |
|---|
| AID773903 | Chemical stability of the compound in Milli-Q water at -30 degC by HPLC analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773894 | Apparent permeability from apical to basolateral side in MDCK cells expressing MDR1 | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773898 | Displacement of [3H]-3-hydroxycyclopent-1-enecarboxylic acid from GHB binding site in Sprague-Dawley rat cerebral cortex after 1 hr by scintillation counting analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID1848977 | Displacement of [3H]NCS-382 from CaMK2alpha in rat brain cortical membrane homogenates measured after 1 hr by TopCount scintillation counting method | | | |
| AID1848978 | Displacement of [3H]HOCPCA from native CaMK2alpha in rat brain cortical membrane homogenates measured after 1 hr by TopCount scintillation counting method | | | |
| AID773902 | Chemical stability of the compound in Milli-Q water assessed as decomposition at room temperature measured on same day by HPLC analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773904 | Displacement of [3H]NCS-382 from GHB binding site in Sprague-Dawley rat brain synaptic membranes after 1 hr by scintillation counting analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID1465898 | Displacement of [3H]NCS-382 from GHB binding site in Sprague-Dawley rat brain synaptosomal membranes after 1 hr by scintillation counting method | 2017 | Journal of medicinal chemistry, 11-09, Volume: 60, Issue:21
| Molecular Hybridization of Potent and Selective γ-Hydroxybutyric Acid (GHB) Ligands: Design, Synthesis, Binding Studies, and Molecular Modeling of Novel 3-Hydroxycyclopent-1-enecarboxylic Acid (HOCPCA) and trans-γ-Hydroxycrotonic Acid (T-HCA) Analogs. |
| AID1848979 | Displacement of [3H]HOCPCA from recombinant rat CaMK2alpha expressed in HEK293T cells measured after 1 hr by liquid scintillation counting method | | | |
| AID773893 | Apparent permeability from basolateral to apical side in MDCK cells expressing MDR1 | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773900 | Chemical stability of the compound in Milli-Q water assessed as decomposition at room temperature after 35 days by HPLC analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773895 | Ratio of drug level in brain to plasma in C57 mouse at 10 mg/kg, po after 30 mins by LC-MS/MS analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| AID773892 | Chemical stability of the compound in Milli-Q water assessed as decomposition at room temperature after 99 days by HPLC analysis | 2013 | Journal of medicinal chemistry, Oct-24, Volume: 56, Issue:20
| New synthesis and tritium labeling of a selective ligand for studying high-affinity γ-hydroxybutyrate (GHB) binding sites. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |