Member | Definition | Class |
acrinathrin | | acrinathrin |
allethrins | | allethrin |
bifenthrin | A carboxylic ester obtained by formal condensation of cis-3-(2-chloro-3,3,3-trifluoroprop-1-enyl)-2,2-dimethylcyclopropanecarboxylic acid and [(2-methyl-1,1'-biphenyl)-3-yl]methanol. | bifenthrin; kappa-bifenthrin |
bifenthrin | A carboxylic ester obtained by formal condensation of the carboxy group of (1R,3R)-3-[(1Z)-2-chloro-3,3,3-trifluoroprop-1-enyl]-2,2-dimethylcyclopropanecarboxylic acid with the hydroxy group of [(2-methyl-1,1'-biphenyl)-3-yl]methanol. | bifenthrin; kappa-bifenthrin |
bioresmethrin | | bioresmethrin |
cyfluthrin | A carboxylic ester obtained by formal condensation between 3-(2,2-dichloroethenyl)-2,2-dimethylcyclopropanecarboxylic acid and (4-fluoro-3-phenoxyphenyl)(hydroxy)acetonitrile. | cyfluthrin |
cyhalothrin | A carboxylic ester obtained by formal condensation between 3-(2-chloro-3,3,3-trifluoroprop-1-en-1-yl)-2,2-dimethylcyclopropanecarboxylic acid and cyano(3-phenoxyphenyl)methanol. | cyhalothrin |
cypermethrin | A carboxylic ester resulting from the formal condensation between 3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropanecarboxylic acid and the alcoholic hydroxy group of hydroxy(3-phenoxyphenyl)acetonitrile. | cypermethrin |
cyphenothrin | | cyphenothrin |
decamethrin | A cyclopropanecarboxylate ester obtained by formal condensation between 3-(2,2-dibromovinyl)-2,2-dimethylcyclopropanecarboxylic acid and cyano(3-phenoxyphenyl)methanol. It is the active insecticide of the proinsecticide tralomethrin. | deltamethrin |
fenpropathrin, (+-)-isomer | A cyclopropanecarboxylate ester obtained by formal condensation between 2,2,3,3-tetramethylcyclopropanecarboxylic acid and cyano(3-phenoxyphenyl)methanol. | fenpropathrin |
fenvalerate | A carboxylic ester obtained by formal condensation between 2-(4-chlorophenyl)-3-methylbutyric acid and cyano(3-phenoxyphenyl)methanol. | fenvalerate |
fluvalinate | | fluvalinate |
permethrin | A cyclopropanecarboxylate ester in which the esterifying alcohol is 3-phenoxybenzyl alcohol and the cyclopropane ring is substituted with a 2,2-dichlorovinyl group and with gem-dimethyl groups. | permethrin |
phenothrin | | phenothrin |
pydrin, (s-(r*,r*))-isomer | | esfenvalerate |
resmethrin | | resmethrin |
tetramethrin | | tetramethrin |
transfluthrin | A carboxylic ester obtained by formal condensation of 3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropanecarboxylic acid and 2,3,5,6-tetrafluorobenzyl alcohol. | transfluthrin |
Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
acetylcholinesterase | Homo sapiens (human) | Potency | 31.7055 | 1 | 1 |
activating transcription factor 6 | Homo sapiens (human) | Potency | 44.6781 | 2 | 10 |
aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 28.1838 | 1 | 1 |
AR protein | Homo sapiens (human) | Potency | 33.9243 | 9 | 52 |
aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 34.2333 | 3 | 7 |
bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 43.1857 | 3 | 24 |
Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 10.2673 | 1 | 3 |
chromobox protein homolog 1 | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 6.9223 | 1 | 5 |
cytochrome P450 2D6 | Homo sapiens (human) | Potency | 18.1543 | 1 | 3 |
cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 12.6354 | 2 | 6 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 25.0424 | 1 | 7 |
DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 39.6705 | 8 | 44 |
estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 36.7849 | 2 | 6 |
estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 45.1310 | 9 | 66 |
euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 35.6383 | 1 | 3 |
farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 32.0500 | 5 | 22 |
G | Vesicular stomatitis virus | Potency | 6.9223 | 1 | 5 |
geminin | Homo sapiens (human) | Potency | 19.8167 | 2 | 3 |
GLI family zinc finger 3 | Homo sapiens (human) | Potency | 26.2216 | 3 | 18 |
glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 37.2720 | 5 | 18 |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 28.3280 | 1 | 3 |
heat shock protein beta-1 | Homo sapiens (human) | Potency | 50.7011 | 2 | 20 |
Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 119.8560 | 1 | 1 |
HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 6.9223 | 1 | 5 |
hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 57.9519 | 1 | 9 |
Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 6.9223 | 1 | 10 |
Interferon beta | Homo sapiens (human) | Potency | 6.9223 | 1 | 5 |
lamin isoform A-delta10 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 14.1254 | 1 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 50.3627 | 3 | 23 |
nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 43.2467 | 1 | 3 |
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 39.5155 | 2 | 15 |
nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 29.9440 | 3 | 34 |
parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 26.5566 | 2 | 2 |
peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 43.1462 | 4 | 24 |
Peroxisome proliferator-activated receptor alpha | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 20.3240 | 3 | 6 |
potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
pregnane X nuclear receptor | Homo sapiens (human) | Potency | 21.8676 | 3 | 37 |
pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 28.3656 | 1 | 11 |
progesterone receptor | Homo sapiens (human) | Potency | 28.6862 | 2 | 16 |
RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 45.2825 | 2 | 30 |
retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 44.1298 | 3 | 19 |
retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 23.5918 | 4 | 24 |
serine-protein kinase ATM isoform a | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
SMAD family member 2 | Homo sapiens (human) | Potency | 23.7692 | 2 | 6 |
SMAD family member 3 | Homo sapiens (human) | Potency | 23.7692 | 2 | 6 |
Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 63.0957 | 1 | 1 |
TDP1 protein | Homo sapiens (human) | Potency | 23.7069 | 2 | 4 |
thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 46.6888 | 3 | 29 |
thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 0.5959 | 2 | 6 |
thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 33.5481 | 4 | 34 |
thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 46.2819 | 1 | 1 |
USP1 protein, partial | Homo sapiens (human) | Potency | 50.3404 | 1 | 3 |
v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 39.3145 | 2 | 10 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 16.1361 | 4 | 8 |
vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 28.3280 | 1 | 3 |