Page last updated: 2024-09-03

ramatroban and diclofenac

ramatroban has been researched along with diclofenac in 5 studies

Compound Research Comparison

Studies
(ramatroban)
Trials
(ramatroban)
Recent Studies (post-2010)
(ramatroban)
Studies
(diclofenac)
Trials
(diclofenac)
Recent Studies (post-2010) (diclofenac)
14210288,8741,8743,616

Protein Interaction Comparison

ProteinTaxonomyramatroban (IC50)diclofenac (IC50)
Aldo-keto reductase family 1 member B10Homo sapiens (human)1.9
Prostaglandin G/H synthase 1 Bos taurus (cattle)0.003
Prostaglandin G/H synthase 1Ovis aries (sheep)1.3376
Interleukin-8Homo sapiens (human)0.008
Prostaglandin G/H synthase 1Homo sapiens (human)0.0415
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)0.5
C-X-C chemokine receptor type 1Homo sapiens (human)0.012
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)0.5
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.5
Prostaglandin G/H synthase 2Homo sapiens (human)0.4165
Prostaglandin G/H synthase 2 Rattus norvegicus (Norway rat)0.5
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.5
Prostaglandin G/H synthase 2Ovis aries (sheep)1.6867
Prostaglandin G/H synthase 2Mus musculus (house mouse)0.0502
Solute carrier family 22 member 6Homo sapiens (human)4
Prostaglandin G/H synthase 1 Rattus norvegicus (Norway rat)0.5
P2Y purinoceptor 12Rattus norvegicus (Norway rat)0.02

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Board, PG; Christ, AN; Clark, AG; Flanagan, JU; Hall, R; Hayes, JD; Hume, DA; Oakley, AJ; Smythe, ML; Weber, JE1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Gyles, SL; Pettipher, R; Townsend, ER; Wettey, F; Xue, L1
Pettipher, R; Townsend, ER; Vinall, SL1
Bachert, C; Holtappels, G; PĂ©rez-Novo, CA; Pettipher, R; Vinall, SL; Xue, L; Zhang, N1

Other Studies

5 other study(ies) available for ramatroban and diclofenac

ArticleYear
Identification and characterisation of new inhibitors for the human hematopoietic prostaglandin D2 synthase.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:2

    Topics: Binding Sites; Drug Evaluation, Preclinical; Enzyme Inhibitors; Glutathione Transferase; Hematopoiesis; Humans; Intramolecular Oxidoreductases; Lipocalins; Models, Molecular; Molecular Conformation; Nocodazole

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A dominant role for chemoattractant receptor-homologous molecule expressed on T helper type 2 (Th2) cells (CRTH2) in mediating chemotaxis of CRTH2+ CD4+ Th2 lymphocytes in response to mast cell supernatants.
    Immunology, 2006, Volume: 119, Issue:3

    Topics: Carbazoles; Cells, Cultured; Chemotaxis, Leukocyte; Culture Media, Conditioned; Cyclooxygenase Inhibitors; Diclofenac; Dose-Response Relationship, Immunologic; Humans; Immunoglobulin E; Lymphocyte Activation; Mast Cells; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Thromboxane; Sulfonamides; Th2 Cells

2006
A paracrine role for chemoattractant receptor-homologous molecule expressed on T helper type 2 cells (CRTH2) in mediating chemotactic activation of CRTH2+ CD4+ T helper type 2 lymphocytes.
    Immunology, 2007, Volume: 121, Issue:4

    Topics: Carbazoles; CD28 Antigens; CD3 Complex; Cells, Cultured; Chemotaxis, Leukocyte; Culture Media, Conditioned; Cyclooxygenase Inhibitors; Cytokines; Diclofenac; Humans; Lymphocyte Activation; Paracrine Communication; Prostaglandin D2; Receptors, Formyl Peptide; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides; Th2 Cells

2007
CRTH2 mediates the activation of human Th2 cells in response to PGD(2) released from IgE/anti-IgE treated nasal polyp tissue.
    Allergy, 2010, Volume: 65, Issue:3

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Antibodies, Anti-Idiotypic; Carbazoles; Chemotaxis, Leukocyte; Diclofenac; Humans; Immunoglobulin E; Lymphocyte Activation; Mast Cells; Nasal Polyps; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides; Th2 Cells

2010