Page last updated: 2024-09-02

2-methylthio-atp and desipramine

2-methylthio-atp has been researched along with desipramine in 2 studies

Compound Research Comparison

Studies
(2-methylthio-atp)
Trials
(2-methylthio-atp)
Recent Studies (post-2010)
(2-methylthio-atp)
Studies
(desipramine)
Trials
(desipramine)
Recent Studies (post-2010) (desipramine)
2650165,775487414

Protein Interaction Comparison

ProteinTaxonomy2-methylthio-atp (IC50)desipramine (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)9.18
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.35
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0034
Alpha-2B adrenergic receptorHomo sapiens (human)0.0003
Alpha-2C adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.35
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.0031
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 6Rattus norvegicus (Norway rat)0.35
Histamine H1 receptorRattus norvegicus (Norway rat)0.0008
Sodium-dependent serotonin transporterHomo sapiens (human)0.1961
5-hydroxytryptamine receptor 7 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5ARattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.35
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0003
Histamine H2 receptorCavia porcellus (domestic guinea pig)3.8
Sodium-dependent dopamine transporter Homo sapiens (human)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.4035
Sodium channel protein type 5 subunit alphaHomo sapiens (human)1.52
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.35
Solute carrier family 22 member 2Rattus norvegicus (Norway rat)10
TransporterRattus norvegicus (Norway rat)7.8

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Najbar-Kaszkiel, AT; Rand, MJ1
Fraga, S; Gonçalves, J; Queiroz, G; Quintas, C1

Other Studies

2 other study(ies) available for 2-methylthio-atp and desipramine

ArticleYear
Effects of P2-receptor agonists on sympathetic neuroeffector transmission in the rat isolated anococcygeus muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:5

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Desipramine; Electric Stimulation; Enzyme Inhibitors; Idazoxan; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; NADP; NG-Nitroarginine Methyl Ester; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Synaptic Transmission; Thionucleotides

1998
The P2Y(1) and P2Y(12) receptors mediate autoinhibition of transmitter release in sympathetic innervated tissues.
    Neurochemistry international, 2009, Volume: 55, Issue:7

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Antidepressive Agents, Tricyclic; Arteries; Blotting, Western; Desipramine; Epididymis; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Neurotransmitter Agents; Norepinephrine; Rats; Rats, Wistar; Receptor Cross-Talk; Receptor, Adenosine A1; Receptors, Adrenergic, alpha-2; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y12; Signal Transduction; Sympathetic Nervous System; Thionucleotides; Vas Deferens

2009
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