Assay ID | Title | Year | Journal | Article |
AID624238 | Antagonists at Human 5-Hydroxytryptamine receptor 5-HT4 | 1998 | Journal of neurochemistry, Jun, Volume: 70, Issue:6
| Cloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminus. |
AID624238 | Antagonists at Human 5-Hydroxytryptamine receptor 5-HT4 | 2000 | British journal of pharmacology, Oct, Volume: 131, Issue:4
| Pharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cells. |
AID1346953 | Human 5-HT4 receptor (5-Hydroxytryptamine receptors) | 2000 | British journal of pharmacology, Feb, Volume: 129, Issue:4
| Isolation of the serotoninergic 5-HT4(e) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell lines. |
AID624238 | Antagonists at Human 5-Hydroxytryptamine receptor 5-HT4 | 2000 | British journal of pharmacology, Jun, Volume: 130, Issue:3
| Exploration of the ligand binding site of the human 5-HT(4) receptor by site-directed mutagenesis and molecular modeling. |
AID1346953 | Human 5-HT4 receptor (5-Hydroxytryptamine receptors) | 2000 | British journal of pharmacology, Oct, Volume: 131, Issue:4
| Pharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cells. |
AID1346953 | Human 5-HT4 receptor (5-Hydroxytryptamine receptors) | 2000 | British journal of pharmacology, Jun, Volume: 130, Issue:3
| Exploration of the ligand binding site of the human 5-HT(4) receptor by site-directed mutagenesis and molecular modeling. |
AID624238 | Antagonists at Human 5-Hydroxytryptamine receptor 5-HT4 | 2004 | British journal of pharmacology, Nov, Volume: 143, Issue:5
| The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo. |
AID1346953 | Human 5-HT4 receptor (5-Hydroxytryptamine receptors) | 1998 | Journal of neurochemistry, Jun, Volume: 70, Issue:6
| Cloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminus. |
AID1346953 | Human 5-HT4 receptor (5-Hydroxytryptamine receptors) | 2004 | British journal of pharmacology, Nov, Volume: 143, Issue:5
| The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo. |
AID624238 | Antagonists at Human 5-Hydroxytryptamine receptor 5-HT4 | 2000 | British journal of pharmacology, Feb, Volume: 129, Issue:4
| Isolation of the serotoninergic 5-HT4(e) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell lines. |
AID6239 | Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligand | 1997 | Journal of medicinal chemistry, Feb-14, Volume: 40, Issue:4
| New esters of 4-amino-5-chloro-2-methoxybenzoic acid as potent agonists and antagonists for 5-HT4 receptors. |
AID5880 | Binding affinity was measured on 5-hydroxytryptamine 3 receptor using [3H]-BRL 43694 as radioligand in rat posterior cortex. | 1997 | Journal of medicinal chemistry, Feb-14, Volume: 40, Issue:4
| New esters of 4-amino-5-chloro-2-methoxybenzoic acid as potent agonists and antagonists for 5-HT4 receptors. |
AID6143 | 5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus and longitudinal muscle of the guinea pig ileum; Inactive up to 10E-5 M | 1997 | Journal of medicinal chemistry, Feb-14, Volume: 40, Issue:4
| New esters of 4-amino-5-chloro-2-methoxybenzoic acid as potent agonists and antagonists for 5-HT4 receptors. |
AID6152 | 5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileum | 1997 | Journal of medicinal chemistry, Feb-14, Volume: 40, Issue:4
| New esters of 4-amino-5-chloro-2-methoxybenzoic acid as potent agonists and antagonists for 5-HT4 receptors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |