Page last updated: 2024-09-04

dk 118 and apomorphine

dk 118 has been researched along with apomorphine in 2 studies

Compound Research Comparison

Studies
(dk 118)
Trials
(dk 118)
Recent Studies (post-2010)
(dk 118)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
7009,205287780

Protein Interaction Comparison

ProteinTaxonomydk 118 (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cannon, JG; Koble, DL; Long, JP; Verimer, T1
Costall, B; Eniojukan, JF; Naylor, RJ1

Other Studies

2 other study(ies) available for dk 118 and apomorphine

ArticleYear
Derivatives of 5-hydroxy-6-methyl-2-aminotetralin.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:7

    Topics: 2-Naphthylamine; Animals; Cats; Dogs; Dopamine; Emetics; Heart; Heart Rate; Humans; Male; Naphthalenes; Rats; Stereotyped Behavior; Structure-Activity Relationship; Synaptic Transmission; Tetrahydronaphthalenes

1980
The mesolimbic nucleus accumbens is critically involved with the mediation of the motor inhibitory and facilitatory effects of dopamine agonists on mouse spontaneous climbing behaviour.
    European journal of pharmacology, 1983, Dec-23, Volume: 96, Issue:3-4

    Topics: Animals; Apomorphine; Behavior, Animal; Dopamine; Dose-Response Relationship, Drug; Female; Mice; Mice, Inbred Strains; Motor Activity; Nucleus Accumbens; Prazosin; Septal Nuclei; Sulpiride; Tetrahydronaphthalenes

1983