Assay ID | Title | Year | Journal | Article |
AID165498 | Compound was tested for agonist activity on rabbit aorta | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID165375 | Tested for the concentration that causes 50% relaxation when contraction in rabbit aorta was induced by 3 x 10 E -8 M of U-46619. | 1990 | Journal of medicinal chemistry, Sep, Volume: 33, Issue:9
| Azulene derivatives: new non-prostanoid thromboxane A2 receptor antagonists. |
AID232743 | Selectivity index for the TXA2 t-receptor was the difference between the IC50 values in the aggregation and contraction assay | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID165497 | Compound was tested for agonist activity on rabbit PRP | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID167793 | Compound was tested for the inhibition U-46619 (3 x10 E -8 M) induced vascular contraction (TXA2 tao receptor) in rabbit thoracic aorta | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID167807 | Displacement of specific binding of [3H]SQ-29,548 to rabbit gel-filtered platelets | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID167790 | Compound was tested for the inhibition U-46619 (3 x10 E -8 M) induced platelet aggregation (TXA2 alpha receptor) in rabbit platelet rich plasma | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID232748 | Selectivity index is the difference between the IC50 values in the aggregation and contraction assays | 1990 | Journal of medicinal chemistry, Sep, Volume: 33, Issue:9
| Azulene derivatives: new non-prostanoid thromboxane A2 receptor antagonists. |
AID92220 | Effect on TXB2 formation of human platelets | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
AID165374 | Tested for the concentration that cause 50% inhibition of the maximum aggregation with rabbit platelet-rich plasma induced by 2.5 x 10 E -6 M of U-46619 | 1990 | Journal of medicinal chemistry, Sep, Volume: 33, Issue:9
| Azulene derivatives: new non-prostanoid thromboxane A2 receptor antagonists. |
AID179228 | Inhibition of U-46619 (3x10E-8 M) induced contraction in rat thoracic aorta | 1993 | Journal of medicinal chemistry, Apr-02, Volume: 36, Issue:7
| Design, synthesis, and pharmacology of 3-substituted sodium azulene-1-sulfonates and related compounds: non-prostanoid thromboxane A2 receptor antagonists. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |