Assay ID | Title | Year | Journal | Article |
AID1092037 | Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assay | 2011 | Journal of agricultural and food chemistry, Apr-13, Volume: 59, Issue:7
| Unique neonicotinoid binding conformations conferring selective receptor interactions. |
AID318725 | Displacement of [3H]ACE from Aplysia AChBP expressed in HEK293S cells by scintillation proximity assay | 2007 | Proceedings of the National Academy of Sciences of the United States of America, May-22, Volume: 104, Issue:21
| Mapping the elusive neonicotinoid binding site. |
AID1092035 | Binding affinity to salt water mollusc Aplysia californica AChBP Y55W mutant assessed as [3H]acetamiprid binding by radioligand binding assay | 2011 | Journal of agricultural and food chemistry, Apr-13, Volume: 59, Issue:7
| Unique neonicotinoid binding conformations conferring selective receptor interactions. |
AID145345 | Potency to displace [3H]IMI binding to Nicotinic acetylcholine receptor from Drosophila head membranes | 2002 | Journal of medicinal chemistry, Jun-20, Volume: 45, Issue:13
| Structural features of azidopyridinyl neonicotinoid probes conferring high affinity and selectivity for mammalian alpha4beta2 and Drosophila nicotinic receptors. |
AID146171 | Potency to displace [3H]nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 immuno-isolated from M10 cells | 2002 | Journal of medicinal chemistry, Jun-20, Volume: 45, Issue:13
| Structural features of azidopyridinyl neonicotinoid probes conferring high affinity and selectivity for mammalian alpha4beta2 and Drosophila nicotinic receptors. |
AID1101289 | Retention time under acidic conditions using H20/MeOH mobile phase containing 0.1% TFA (1:1) by HPLC method | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1101293 | Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1101290 | Retention time under neutral conditions using H20/MeOH (1:1) mobile phase by HPLC method | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1092036 | Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand binding assay | 2011 | Journal of agricultural and food chemistry, Apr-13, Volume: 59, Issue:7
| Unique neonicotinoid binding conformations conferring selective receptor interactions. |
AID220121 | Inhibition of [3H](-)-nicotine binding to recombinant rat alpha4-beta2 nAChR. | 1999 | Journal of medicinal chemistry, Jun-17, Volume: 42, Issue:12
| Novel and potent 6-chloro-3-pyridinyl ligands for the alpha4beta2 neuronal nicotinic acetylcholine receptor. |
AID1101288 | Retention time under basic conditions using 20 mM Na2HPO4 (pH9.9)/MeOH (1:1) mobile phase by HPLC method | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID318726 | Displacement of [3H]EPI from Aplysia AChBP expressed in HEK293S cells by scintillation proximity assay | 2007 | Proceedings of the National Academy of Sciences of the United States of America, May-22, Volume: 104, Issue:21
| Mapping the elusive neonicotinoid binding site. |
AID1101291 | Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylcholine receptor subunits | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1101292 | Inhibition of [3H]nicotine binding to alpha3 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells co-expressing beta2beta4alpha5 Nicotinic acetylcholine receptor subunits | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID145850 | Selectivity ratio of Ki of Nicotinic acetylcholine receptor of Drosophila to Nicotinic acetylcholine receptor alpha4-beta2 | 2002 | Journal of medicinal chemistry, Jun-20, Volume: 45, Issue:13
| Structural features of azidopyridinyl neonicotinoid probes conferring high affinity and selectivity for mammalian alpha4beta2 and Drosophila nicotinic receptors. |
AID1101298 | Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptor | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1092034 | Binding affinity to freshwater snail Lymnaea stagnalis AChBP assessed as [3H]EPI binding by radioligand binding assay | 2011 | Journal of agricultural and food chemistry, Apr-13, Volume: 59, Issue:7
| Unique neonicotinoid binding conformations conferring selective receptor interactions. |
AID1101296 | Toxicity against Musca domestica (house fly) dosed with compound through intra-thoracic injection pre-treated with 100 ug/g metabolic detoxification inhibitor O-propyl O-(2-propynyl)phenylphosphonate | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1101295 | Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta1 nicotinic acetylcholine receptor subunits | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
AID1091945 | Insecticidal activity against Nephotettix cincticeps (green rice leafhopper) assessed as mortality measured after 4 days | 2011 | Journal of agricultural and food chemistry, Apr-13, Volume: 59, Issue:7
| Discovery of imidacloprid and further developments from strategic molecular designs. |
AID1101297 | Toxicity in ip dosed Mus musculus (mouse) | 2000 | Journal of agricultural and food chemistry, Dec, Volume: 48, Issue:12
| Neonicotinoid insecticides: molecular features conferring selectivity for insect versus mammalian nicotinic receptors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |