Assay ID | Title | Year | Journal | Article |
AID309785 | Half life in Sprague-Dawley rat at 20 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309775 | Mean residential time (0 to infinity) in Sprague-Dawley rat at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309774 | Mean residential time (0 to infinity) in Sprague-Dawley rat at 1.25 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309772 | AUC (0 to infinity) in Sprague-Dawley rat at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309778 | Clearance (0 to infinity) in Sprague-Dawley rat at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309796 | Half life in cynomolgus monkey at 1 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309764 | Aqueous solubility at pH 6.8 | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309787 | Drug level in cynomolgus monkey serum at 5 mg/kg, iv after 1 hr | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309769 | Drug level in Sprague-Dawley rat serum at 5 mg/kg, iv after 2 hrs | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309788 | AUC (0 to infinity) in cynomolgus monkey at 1 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309773 | AUC (0 to infinity) in Sprague-Dawley rat at 20 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309771 | AUC (0 to infinity) in Sprague-Dawley rat at 1.25 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309770 | Drug level in Sprague-Dawley rat serum at 20 mg/kg, iv after 2 hrs | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309766 | Toxicity in mouse assessed as lethal effect at 100 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309792 | Clearance (0 to infinity) in cynomolgus monkey at 1 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309780 | Volume of distribution at steady state (0 to infinity) in Sprague-Dawley rat at 1.25 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309791 | Mean residential time (0 to infinity) in cynomolgus monkey at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309789 | AUC (0 to infinity) in cynomolgus monkey at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309768 | Drug level in Sprague-Dawley rat serum at 1.25 mg/kg, iv after 2 hrs | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309781 | Volume of distribution at steady state (0 to infinity) in Sprague-Dawley rat at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309784 | Half life in Sprague-Dawley rat at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309786 | Drug level in cynomolgus monkey serum at 1 mg/kg, iv after 1 hr | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309790 | Mean residential time (0 to infinity) in cynomolgus monkey at 1 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309793 | Clearance (0 to infinity) in cynomolgus monkey at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309762 | Inhibition of Pseudomonas aeruginosa PAM1723 MexAB-OprM assessed as drug level required to decrease MIC of levofloxacin in presence of 0.125% HAS | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309761 | Inhibition of Pseudomonas aeruginosa PAM1723 MexAB-OprM assessed as drug level required to decrease MIC of levofloxacin | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309763 | Inhibition of Pseudomonas aeruginosa PAM1723 MexAB-OprM assessed as drug level required to decrease MIC of aztreonam | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309776 | Mean residential time (0 to infinity) in Sprague-Dawley rat at 20 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309797 | Half life in cynomolgus monkey at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309794 | Volume of distribution at steady state (0 to infinity) in cynomolgus monkey at 1 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309777 | Clearance (0 to infinity) in Sprague-Dawley rat at 1.25 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309795 | Volume of distribution at steady state (0 to infinity) in cynomolgus monkey at 5 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309779 | Clearance (0 to infinity) in Sprague-Dawley rat at 20 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309782 | Volume of distribution at steady state (0 to infinity) in Sprague-Dawley rat at 20 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
AID309783 | Half life in Sprague-Dawley rat at 1.25 mg/kg, iv | 2007 | Bioorganic & medicinal chemistry, Nov-15, Volume: 15, Issue:22
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |