Page last updated: 2024-09-02

sr 95531 and orlistat

sr 95531 has been researched along with orlistat in 2 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(orlistat)
Trials
(orlistat)
Recent Studies (post-2010) (orlistat)
61002091,432274539

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)orlistat (IC50)
Phosphatidylserine lipase ABHD16AHomo sapiens (human)0.1
Pancreatic triacylglycerol lipaseSus scrofa (pig)0.4214
Lipoprotein lipaseHomo sapiens (human)0.066
Cytochrome P450 3A4Homo sapiens (human)0.42
Hepatic triacylglycerol lipaseHomo sapiens (human)0.003
Pancreatic triacylglycerol lipaseHomo sapiens (human)0.3253
Translocator proteinRattus norvegicus (Norway rat)1
Cytochrome P450 2C19Homo sapiens (human)0.42
Kappa-type opioid receptorMus musculus (house mouse)0.1903
Fatty acid synthaseHomo sapiens (human)2.99
Fatty-acid amide hydrolase 1Rattus norvegicus (Norway rat)0.01
Platelet-activating factor acetylhydrolaseHomo sapiens (human)0.05
Diacylglycerol lipase-alphaMus musculus (house mouse)0.02
Lysophosphatidylserine lipase ABHD12Homo sapiens (human)0.1682
Diacylglycerol lipase-betaHomo sapiens (human)0.24
Monoacylglycerol lipase ABHD6Homo sapiens (human)0.03
Acyl-protein thioesterase 2Rattus norvegicus (Norway rat)0.17
Diacylglycerol lipase-alphaHomo sapiens (human)0.2677
Endothelial lipaseHomo sapiens (human)0.006

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Huang, GZ; Woolley, CS1
Conde, K; Fabelo, C; Fischer, D; Goethel, J; Hur, J; Ingraham, HA; Krause, WC; Meza, C; Propst, R; Wagner, EJ1

Other Studies

2 other study(ies) available for sr 95531 and orlistat

ArticleYear
Estradiol acutely suppresses inhibition in the hippocampus through a sex-specific endocannabinoid and mGluR-dependent mechanism.
    Neuron, 2012, Jun-07, Volume: 74, Issue:5

    Topics: Animals; Benzodioxoles; Benzoxazines; Biophysics; CA1 Region, Hippocampal; Cannabinoid Receptor Modulators; Castration; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estradiol; Estrogens; Excitatory Amino Acid Agents; Female; GABA Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Lactones; Male; Morpholines; NAD; Naphthalenes; Neural Inhibition; Neurons; Orlistat; Patch-Clamp Techniques; Phenols; Piperidines; Pyrazoles; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate

2012
Testosterone Rapidly Augments Retrograde Endocannabinoid Signaling in Proopiomelanocortin Neurons to Suppress Glutamatergic Input from Steroidogenic Factor 1 Neurons via Upregulation of Diacylglycerol Lipase-α.
    Neuroendocrinology, 2017, Volume: 105, Issue:4

    Topics: Action Potentials; Animals; Cerebral Cortex; Endocannabinoids; Energy Intake; Enzyme Inhibitors; Estradiol; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Glutamic Acid; Guinea Pigs; Lactones; Lipoprotein Lipase; Male; Neural Pathways; Neurons; Orlistat; Pro-Opiomelanocortin; Pyridazines; Signal Transduction; Steroidogenic Factor 1; Testosterone; Up-Regulation

2017