Page last updated: 2024-09-04

abiraterone and niraparib

abiraterone has been researched along with niraparib in 1 studies

Compound Research Comparison

Studies
(abiraterone)
Trials
(abiraterone)
Recent Studies (post-2010)
(abiraterone)
Studies
(niraparib)
Trials
(niraparib)
Recent Studies (post-2010) (niraparib)
9429785421246209

Protein Interaction Comparison

ProteinTaxonomyabiraterone (IC50)niraparib (IC50)
Poly [ADP-ribose] polymerase tankyrase-1Homo sapiens (human)1.7564
Poly [ADP-ribose] polymerase 1Homo sapiens (human)0.0278
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0021
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0021
Protein mono-ADP-ribosyltransferase PARP14Homo sapiens (human)1.7378
Protein mono-ADP-ribosyltransferase PARP10Homo sapiens (human)2.6153
Protein mono-ADP-ribosyltransferase PARP12Homo sapiens (human)0.4367
Poly [ADP-ribose] polymerase tankyrase-2Homo sapiens (human)5.1293
Poly [ADP-ribose] polymerase 2Homo sapiens (human)0.2306
Protein mono-ADP-ribosyltransferase PARP4Homo sapiens (human)0.4076
Protein mono-ADP-ribosyltransferase PARP3Homo sapiens (human)0.3797

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Bradic, B; Chi, KN; De Meulder, M; Espina, BM; Francis, P; Graff, JN; Hayreh, V; Hazra, A; Lattouf, JB; Mamidi, RNVS; Posadas, EM; Rezazadeh Kalebasty, A; Saad, F; Shore, ND; Yu, A; Zhu, E1

Trials

1 trial(s) available for abiraterone and niraparib

ArticleYear
Niraparib with androgen receptor-axis-targeted therapy in patients with metastatic castration-resistant prostate cancer: safety and pharmacokinetic results from a phase 1b study (BEDIVERE).
    Cancer chemotherapy and pharmacology, 2021, Volume: 88, Issue:1

    Topics: Aged; Aged, 80 and over; Androstenes; Antineoplastic Combined Chemotherapy Protocols; Humans; Indazoles; Male; Middle Aged; Piperidines; Poly(ADP-ribose) Polymerase Inhibitors; Prednisone; Prostatic Neoplasms, Castration-Resistant; Receptors, Androgen; Thiohydantoins

2021
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