A thyroid hormone receptor beta that is encoded in the genome of rat. [OMA:P18113, PRO:DNx]
Nuclear receptor subfamily 1 group A member 2;
c-erbA-2;
c-erbA-beta
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 2 (33.33) | 18.7374 |
1990's | 4 (66.67) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
theophylline | Rattus norvegicus (Norway rat) | Ki | 14.0000 | 1 | 1 |
amiodarone | Rattus norvegicus (Norway rat) | IC50 | 200.0000 | 1 | 1 |
3,3',5-triiodothyroacetic acid | Rattus norvegicus (Norway rat) | IC50 | 0.0001 | 1 | 1 |
triiodothyronine | Rattus norvegicus (Norway rat) | IC50 | 0.0031 | 1 | 2 |
dextrothyroxine | Rattus norvegicus (Norway rat) | IC50 | 0.0350 | 1 | 1 |
1-methylxanthine | Rattus norvegicus (Norway rat) | Ki | 9.0000 | 1 | 1 |
n(6)-benzyladenosine | Rattus norvegicus (Norway rat) | Ki | 4.4500 | 1 | 1 |
5'-n-methylcarboxamideadenosine | Rattus norvegicus (Norway rat) | Ki | 1.0840 | 1 | 2 |
desethylamiodarone | Rattus norvegicus (Norway rat) | IC50 | 27.0000 | 1 | 1 |
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosine | Rattus norvegicus (Norway rat) | Ki | 0.0540 | 1 | 2 |
di-n-desethylamiodarone | Rattus norvegicus (Norway rat) | IC50 | 19.0000 | 1 | 1 |
1,3-dipropylxanthine | Rattus norvegicus (Norway rat) | Ki | 0.7000 | 1 | 1 |
adenosine-5'-(n-ethylcarboxamide) | Rattus norvegicus (Norway rat) | Ki | 0.0630 | 1 | 2 |
n(6)-cyclopentyladenosine | Rattus norvegicus (Norway rat) | Ki | 0.0059 | 1 | 1 |
adenosine-5'-(N-propyl)carboxamide | Rattus norvegicus (Norway rat) | Ki | 1.2400 | 1 | 2 |
cgs 23425 | Rattus norvegicus (Norway rat) | IC50 | 0.0002 | 1 | 1 |
n-cyclopropyl adenosine-5'-carboxamide | Rattus norvegicus (Norway rat) | Ki | 0.0630 | 1 | 2 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pralidoxime iodide | Rattus norvegicus (Norway rat) | Kr | 1,100,000,000.0000 | 1 | 1 |