Page last updated: 2024-08-07 16:04:50

Thyroid hormone receptor beta

A thyroid hormone receptor beta that is encoded in the genome of rat. [OMA:P18113, PRO:DNx]

Synonyms

Nuclear receptor subfamily 1 group A member 2;
c-erbA-2;
c-erbA-beta

Research

Bioassay Publications (6)

TimeframeStudies on this Protein(%)All Drugs %
pre-19902 (33.33)18.7374
1990's4 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (18)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
theophyllineRattus norvegicus (Norway rat)Ki14.000011
amiodaroneRattus norvegicus (Norway rat)IC50200.000011
3,3',5-triiodothyroacetic acidRattus norvegicus (Norway rat)IC500.000111
triiodothyronineRattus norvegicus (Norway rat)IC500.003112
dextrothyroxineRattus norvegicus (Norway rat)IC500.035011
1-methylxanthineRattus norvegicus (Norway rat)Ki9.000011
n(6)-benzyladenosineRattus norvegicus (Norway rat)Ki4.450011
5'-n-methylcarboxamideadenosineRattus norvegicus (Norway rat)Ki1.084012
desethylamiodaroneRattus norvegicus (Norway rat)IC5027.000011
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosineRattus norvegicus (Norway rat)Ki0.054012
di-n-desethylamiodaroneRattus norvegicus (Norway rat)IC5019.000011
1,3-dipropylxanthineRattus norvegicus (Norway rat)Ki0.700011
adenosine-5'-(n-ethylcarboxamide)Rattus norvegicus (Norway rat)Ki0.063012
n(6)-cyclopentyladenosineRattus norvegicus (Norway rat)Ki0.005911
adenosine-5'-(N-propyl)carboxamideRattus norvegicus (Norway rat)Ki1.240012
cgs 23425Rattus norvegicus (Norway rat)IC500.000211
n-cyclopropyl adenosine-5'-carboxamideRattus norvegicus (Norway rat)Ki0.063012

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pralidoxime iodideRattus norvegicus (Norway rat)Kr1,100,000,000.000011